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7ALF
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BU of 7alf by Molmil
The dimethylated RSL - sulfonato-calix[8]arene complex, P3 form, acetate pH 4.0
分子名称: Fucose-binding lectin protein, GLYCEROL, beta-D-fructopyranose, ...
著者Ramberg, K, Engilberge, S, Crowley, P.B.
登録日2020-10-06
公開日2021-04-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.261 Å)
主引用文献Facile Fabrication of Protein-Macrocycle Frameworks.
J.Am.Chem.Soc., 143, 2021
8Q7P
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BU of 8q7p by Molmil
Tau - AD-MIA8 (intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-16
公開日2023-08-30
最終更新日2024-01-24
実験手法ELECTRON MICROSCOPY (3.28 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q3U
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BU of 8q3u by Molmil
Crystal structure of a fentanyl derivative in complex with human CA VII
分子名称: Carbonic anhydrase 7, GLYCEROL, ZINC ION, ...
著者Alterio, V, Di Fiore, A, De Simone, G.
登録日2023-08-04
公開日2023-09-20
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Discovery of a novel series of potent carbonic anhydrase inhibitors with selective affinity for mu Opioid receptor for Safer and long-lasting analgesia.
Eur.J.Med.Chem., 260, 2023
8PYN
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BU of 8pyn by Molmil
Human IGF1R with inhibitor 56
分子名称: 5,5-dimethyl-1-(1H-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfonyl)phenyl]imidazolidine-2,4-dione, CADMIUM ION, Insulin-like growth factor 1 receptor beta chain, ...
著者Dreyer, M.K, Wang, J, Elkins, J.M.
登録日2023-07-25
公開日2023-09-20
実験手法X-RAY DIFFRACTION (1.71 Å)
主引用文献Human IGF1R with inhibitor 56
To Be Published
8Q8M
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BU of 8q8m by Molmil
Tau - AD-PHF long crossover
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-18
公開日2023-09-20
最終更新日2024-01-24
実験手法ELECTRON MICROSCOPY (2.95 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q98
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BU of 8q98 by Molmil
Tau - CTE-MIA8 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-20
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (1.75 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q2L
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BU of 8q2l by Molmil
Tau - AD-MIA4
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-02
公開日2023-09-20
最終更新日2024-01-24
実験手法ELECTRON MICROSCOPY (2.2 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8PYM
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BU of 8pym by Molmil
Human IGF1R with inhibitor 54
分子名称: 5,5-dimethyl-1-(1H-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dione, CADMIUM ION, Insulin-like growth factor 1 receptor beta chain, ...
著者Dreyer, M.K, Wang, J, Elkins, J.M.
登録日2023-07-25
公開日2023-09-20
実験手法X-RAY DIFFRACTION (2.652 Å)
主引用文献Human IGF1R with inhibitor 54
To Be Published
8Q97
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BU of 8q97 by Molmil
Tau - CTE-MIA9 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-20
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (2.99 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q2D
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BU of 8q2d by Molmil
Crystal structure of the E. coli PqiC Lipoprotein residues 17-187
分子名称: Intermembrane transport lipoprotein PqiC
著者Cooper, B.F, Knowles, T.J.
登録日2023-08-02
公開日2023-09-20
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献An octameric PqiC toroid stabilises the outer-membrane interaction of the PqiABC transport system.
Embo Rep., 25, 2024
8Q9D
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BU of 8q9d by Molmil
Tau - CTE-MIA15 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-20
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (3.16 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8PM3
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BU of 8pm3 by Molmil
Crystal structure of MAP2K6 with a covalent compound GCL94
分子名称: Dual specificity mitogen-activated protein kinase kinase 6, ~{N}-[3-(2-azanylpyridin-4-yl)phenyl]propanamide
著者Wang, G.Q, Seidler, N, Roehm, S, Gehringer, M, Knapp, S, Structural Genomics Consortium (SGC)
登録日2023-06-28
公開日2023-09-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of MAP2K6 with a covalent compound GCL94
To Be Published
8Q2C
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BU of 8q2c by Molmil
Crystal structure of the E. coli PqiC Lipoprotein
分子名称: Intermembrane transport lipoprotein PqiC
著者Cooper, B.F, Ratkeviciute, G.R, Knowles, T.J.
登録日2023-08-02
公開日2023-09-20
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (3.21 Å)
主引用文献An octameric PqiC toroid stabilises the outer-membrane interaction of the PqiABC transport system.
Embo Rep., 25, 2024
8PVO
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BU of 8pvo by Molmil
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with allosteric compound FG5
分子名称: 1,2-ETHANEDIOL, 2-[1-(1,3-benzothiazol-6-ylsulfonyl)piperidin-4-yl]-~{N}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine, Casein kinase II subunit alpha, ...
著者Kraemer, A, Greco, F, Knapp, S, Structural Genomics Consortium (SGC)
登録日2023-07-18
公開日2023-09-20
最終更新日2024-08-07
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Synthesis and evaluation of chemical linchpins for highly selective CK2 alpha targeting.
Eur.J.Med.Chem., 276, 2024
8Q8F
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BU of 8q8f by Molmil
Tau - AD-LIA5 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-18
公開日2023-09-20
最終更新日2024-01-24
実験手法ELECTRON MICROSCOPY (2.93 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q8V
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BU of 8q8v by Molmil
Tau - CTE-MIA3
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-18
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q8L
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BU of 8q8l by Molmil
Tau - AD-LIA7 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-18
公開日2023-09-20
最終更新日2024-01-24
実験手法ELECTRON MICROSCOPY (3.04 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q9C
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BU of 8q9c by Molmil
Tau - CTE-MIA14 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-20
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q8U
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BU of 8q8u by Molmil
Tau - CTE-MIA1 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-18
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q8W
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BU of 8q8w by Molmil
Tau - CTE-MIA4 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-19
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (2.85 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q3O
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BU of 8q3o by Molmil
Bacterial transcription termination factor Rho + pppGpp
分子名称: MAGNESIUM ION, Transcription termination factor Rho, guanosine 5'-(tetrahydrogen triphosphate) 3'-(trihydrogen diphosphate)
著者Said, N, Hilal, T, Wahl, M.C.
登録日2023-08-04
公開日2023-09-27
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Transcription termination factor rho polymerizes under stress.
Biorxiv, 2023
8Q8Y
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BU of 8q8y by Molmil
Tau - CTE-MIA6 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-19
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (2.88 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8PH7
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BU of 8ph7 by Molmil
X-ray structure of the adduct formed upon reaction of Lysozyme with [Ru2Cl(DPhF)(O2CCH3)3] in condition A
分子名称: Lysozyme C, SODIUM ION, SUCCINIC ACID, ...
著者Teran, A, Ferraro, G, Merlino, A.
登録日2023-06-19
公開日2023-09-13
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.406 Å)
主引用文献Steric hindrance and charge influence on the cytotoxic activity and protein binding properties of diruthenium complexes.
Int.J.Biol.Macromol., 253, 2023
8Q9E
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BU of 8q9e by Molmil
Tau - CTE-MIA18 (tau intermediate amyloid)
分子名称: Isoform Tau-D of Microtubule-associated protein tau
著者Lovestam, S, Li, D, Scheres, S.H.W, Goedert, M.
登録日2023-08-20
公開日2023-09-20
最終更新日2024-01-17
実験手法ELECTRON MICROSCOPY (2.97 Å)
主引用文献Disease-specific tau filaments assemble via polymorphic intermediates.
Nature, 625, 2024
8Q0P
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BU of 8q0p by Molmil
Crystal Structure of an N-terminal Domain of Variant Surface Glycoprotein 21 (VSG21) of Trypanosome brucei brucei Lister 427
分子名称: Variant surface glycoprotein MITat 1.21
著者Zeelen, J.P, Stebbins, C.E.
登録日2023-07-28
公開日2023-09-13
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献A structural classification of the variant surface glycoproteins of the African trypanosomey.
Plos Negl Trop Dis, 17, 2023

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件を2024-08-21に公開中

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