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2H1W
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Crystal structure of the His183Ala mutant variant of Bacillus subtilis ferrochelatase
分子名称: FE (II) ION, Ferrochelatase, MAGNESIUM ION
著者Hansson, M.D, Karlberg, T, Arys Rahardja, M, Al-Karadaghi, S, Hansson, M.
登録日2006-05-17
公開日2007-01-16
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Amino Acid Residues His183 and Glu264 in Bacillus subtilis Ferrochelatase Direct and Facilitate the Insertion of Metal Ion into Protoporphyrin IX
Biochemistry, 46, 2007
2H4X
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Human bisphosphoglycerate mutase complex with 3-phosphoglycerate with crystal growth 90 days
分子名称: 3-PHOSPHOGLYCERIC ACID, Bisphosphoglycerate mutase
著者Wang, Y, Gong, W.
登録日2006-05-25
公開日2006-10-24
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Seeing the process of histidine phosphorylation in human bisphosphoglycerate mutase.
J.Biol.Chem., 281, 2006
2H5S
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SA2-13 penam sulfone complexed to wt SHV-1 beta-lactamase
分子名称: (3R)-4-[(4-CARBOXYBUTANOYL)OXY]-N-[(1E)-3-OXOPROP-1-EN-1-YL]-3-SULFINO-D-VALINE, CYCLOHEXYL-HEXYL-BETA-D-MALTOSIDE, SHV-1 beta-lactamase
著者van den Akker, F, Padayatti, P.S.
登録日2006-05-27
公開日2006-10-17
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.28 Å)
主引用文献Rational Design of a beta-Lactamase Inhibitor Achieved via Stabilization of the trans-Enamine Intermediate: 1.28 A Crystal Structure of wt SHV-1 Complex with a Penam Sulfone.
J.Am.Chem.Soc., 128, 2006
2GS4
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The crystal structure of the E.coli stress protein YciF.
分子名称: Protein yciF
著者Hindupur, A, Liu, D, Zhao, Y, Bellamy, H.D, White, M.A, Fox, R.O.
登録日2006-04-25
公開日2006-10-17
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The crystal structure of the E. coli stress protein YciF.
Protein Sci., 15, 2006
4LU3
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The crystal structure of the human carbonic anhydrase XIV
分子名称: 5-ACETAMIDO-1,3,4-THIADIAZOLE-2-SULFONAMIDE, Carbonic anhydrase 14, GLYCEROL, ...
著者Alterio, V, De Simone, G, Monti, S.M.
登録日2013-07-24
公開日2014-01-01
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The structural comparison between membrane-associated human carbonic anhydrases provides insights into drug design of selective inhibitors.
Biopolymers, 101, 2014
4CCB
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Structure of the Human Anaplastic Lymphoma Kinase in Complex with 3-((R)-1-(5-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl)ethoxy)-5-(5-methyl-1H- pyrazol-4-yl)pyridin-2-amine
分子名称: 3-[(1R)-1-[5-fluoranyl-2-(1,2,3-triazol-2-yl)phenyl]ethoxy]-5-(3-methyl-1H-pyrazol-4-yl)pyridin-2-amine, ALK TYROSINE KINASE RECEPTOR
著者McTigue, M, Deng, Y, Liu, W, Brooun, A, Stewart, A.
登録日2013-10-21
公開日2014-01-29
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献The Design of Potent and Selective Inhibitors to Overcome Clinical Alk Mutations Resistant to Crizotinib.
J.Med.Chem., 57, 2014
2GQF
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Crystal structure of flavoprotein HI0933 from Haemophilus influenzae Rd
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, Hypothetical protein HI0933, SULFATE ION
著者Mulichak, A.M, Patskovsky, Y, Keefe, L.J, Almo, S.C, Burley, S.K, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2006-04-20
公開日2006-05-30
最終更新日2021-02-03
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of hypothetical flavoprotein HI0933 from Haemophilus influenzae Rd.
To be Published
2H2D
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The Structural Basis for Sirtuin Substrate Affinity
分子名称: Cellular tumor antigen p53 peptide, NAD-dependent deacetylase, ZINC ION
著者Cosgrove, M.S, Wolberger, C.
登録日2006-05-18
公開日2006-09-19
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献On the Structural Basis of Sirtuin Substrate Affinity
Biochemistry, 45, 2006
2H2F
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The Structural basis for Sirtuin Substrate affinity
分子名称: Cellular tumor antigen p53, NAD-dependent deacetylase, ZINC ION
著者Cosgrove, M.S, Wolberger, C.
登録日2006-05-18
公開日2006-12-05
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The structural basis of sirtuin substrate affinity
Biochemistry, 45, 2006
2H2J
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Structure of Rubisco LSMT bound to Sinefungin and Monomethyllysine
分子名称: N-METHYL-LYSINE, Ribulose-1,5 bisphosphate carboxylase/oxygenase large subunit N-methyltransferase, SINEFUNGIN
著者Couture, J.F, Hauk, G, Trievel, R.C.
登録日2006-05-18
公開日2006-05-30
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Catalytic Roles for Carbon-Oxygen Hydrogen Bonding in SET Domain Lysine Methyltransferases.
J.Biol.Chem., 281, 2006
2H55
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Structure of human Hsp90-alpha bound to the potent water soluble inhibitor PU-DZ8
分子名称: 2-FLUORO-8-[(6-IODO-1,3-BENZODIOXOL-5-YL)METHYL]-9-[3-(ISOPROPYLAMINO)PROPYL]-9H-PURIN-6-AMINE, Heat shock protein HSP 90-alpha 4
著者Immormino, R.M, Gewirth, D.T.
登録日2006-05-25
公開日2006-10-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and quantum chemical studies of 8-aryl-sulfanyl adenine class Hsp90 inhibitors.
J.Med.Chem., 49, 2006
4CCO
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BU of 4cco by Molmil
60S ribosomal protein L8 histidine hydroxylase (NO66 S373C) in complex with Mn(II), N-oxalylglycine (NOG) and 60S ribosomal protein L8 (RPL8 G214C) peptide fragment (complex-3)
分子名称: 1,2-ETHANEDIOL, 60S RIBOSOMAL PROTEIN L8, BIFUNCTIONAL LYSINE-SPECIFIC DEMETHYLASE AND HISTIDYL-HYDROXYLASE NO66, ...
著者Chowdhury, R, Schofield, C.J.
登録日2013-10-23
公開日2014-05-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Ribosomal oxygenases are structurally conserved from prokaryotes to humans.
Nature, 510, 2014
2PSM
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Crystal structure of Interleukin 15 in complex with Interleukin 15 receptor alpha
分子名称: BENZAMIDINE, Interleukin-15, Interleukin-15 receptor alpha chain
著者Olsen, S.K, Murayama, K, Kishishita, S, Kukimoto-Niino, M, Terada, T, Shirouzu, M, Ota, N, Kanagawa, O, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-05-07
公開日2007-11-06
最終更新日2021-08-18
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Crystal Structure of the Interleukin-15{middle dot}Interleukin-15 Receptor {alpha} Complex: INSIGHTS INTO TRANS AND CIS PRESENTATION
J.Biol.Chem., 282, 2007
4C2H
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BU of 4c2h by Molmil
Crystal structure of the CtpB(V118Y) mutant
分子名称: CARBOXY-TERMINAL PROCESSING PROTEASE CTPB
著者Mastny, M, Heuck, A, Kurzbauer, R, Clausen, T.
登録日2013-08-17
公開日2013-12-04
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Ctpb Assembles a Gated Protease Tunnel Regulating Cell-Cell Signaling During Spore Formation in Bacillus Subtilis.
Cell(Cambridge,Mass.), 155, 2013
2KMB
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COMPLEX OF 3'-NEUAC-LEWIS-X WITH A SELECTIN-LIKE MUTANT OF MANNOSE-BINDING PROTEIN A
分子名称: CALCIUM ION, CHLORIDE ION, MANNOSE-BINDING PROTEIN-A, ...
著者Ng, K.K.-S, Weis, W.I.
登録日1996-11-07
公開日1997-02-12
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of a selectin-like mutant of mannose-binding protein complexed with sialylated and sulfated Lewis(x) oligosaccharides.
Biochemistry, 36, 1997
4CCM
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60S ribosomal protein L8 histidine hydroxylase (NO66) in complex with Mn(II), N-oxalylglycine (NOG) and 60S ribosomal protein L8 (RPL8 G220C) peptide fragment (complex-1)
分子名称: 1,2-ETHANEDIOL, 60S RIBOSOMAL PROTEIN L8, BIFUNCTIONAL LYSINE-SPECIFIC DEMETHYLASE AND HISTIDYL-HYDROXYLASE NO66, ...
著者Chowdhury, R, Schofield, C.J.
登録日2013-10-23
公開日2014-05-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Ribosomal oxygenases are structurally conserved from prokaryotes to humans.
Nature, 510, 2014
4CD0
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BU of 4cd0 by Molmil
Structure of L1196M Mutant Human Anaplastic Lymphoma Kinase in Complex with 2-(5-(6-amino-5-((R)-1-(5-fluoro-2-(2H-1,2,3-triazol-2- yl)phenyl)ethoxy)pyridin-3-yl)-4-methylthiazol-2-yl)propane-1,2-diol
分子名称: (2R)-2-[5-(6-amino-5-{(1R)-1-[2-(1,3-dihydro-2H-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diol, ALK TYROSINE KINASE RECEPTOR
著者McTigue, M, Deng, Y, Liu, W, Brooun, A, Stewart, A.
登録日2013-10-29
公開日2014-01-29
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献The Design of Potent and Selective Inhibitors to Overcome Clinical Alk Mutations Resistant to Crizotinib.
J.Med.Chem., 57, 2014
2GW8
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Structure of the PII signal transduction protein of Neisseria meningitidis at 1.85 resolution
分子名称: PII signal transduction protein
著者Nichols, C.E, Sainsbury, S, Berrow, N.S, Alderton, D, Stammers, D.K, Owens, R.J, Oxford Protein Production Facility (OPPF)
登録日2006-05-04
公開日2006-06-13
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structure of the P(II) signal transduction protein of Neisseria meningitidis at 1.85 A resolution.
Acta Crystallogr.,Sect.F, 62, 2006
2GX0
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Crystal structural and functional analysis of GFP-like fluorescent protein
分子名称: fluorescent protein Dronpa
著者Hwang, K.Y, Nam, K.-H, Park, S.-Y, Sugiyama, K.
登録日2006-05-08
公開日2007-05-08
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural characterization of the photoswitchable fluorescent protein Dronpa-C62S
Biochem.Biophys.Res.Commun., 354, 2007
2HDH
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BIOCHEMICAL CHARACTERIZATION AND STRUCTURE DETERMINATION OF HUMAN HEART SHORT CHAIN L-3-HYDROXYACYL COA DEHYDROGENASE PROVIDE INSIGHT INTO CATALYTIC MECHANISM
分子名称: L-3-HYDROXYACYL COA DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Barycki, J.J, Bratt, J.M, Banaszak, L.J.
登録日1998-12-04
公開日1999-05-12
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Biochemical characterization and crystal structure determination of human heart short chain L-3-hydroxyacyl-CoA dehydrogenase provide insights into catalytic mechanism.
Biochemistry, 38, 1999
2H21
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Structure of Rubisco LSMT bound to AdoMet
分子名称: Ribulose-1,5 bisphosphate carboxylase/oxygenase, S-ADENOSYLMETHIONINE
著者Couture, J.F, Hauk, G, Trievel, R.C.
登録日2006-05-17
公開日2006-05-30
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Catalytic Roles for Carbon-Oxygen Hydrogen Bonding in SET Domain Lysine Methyltransferases.
J.Biol.Chem., 281, 2006
2GNK
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GLNK, A SIGNAL PROTEIN FROM E. COLI
分子名称: ADENOSINE-5'-TRIPHOSPHATE, PROTEIN (NITROGEN REGULATORY PROTEIN)
著者Xu, Y, Cheah, E, Carr, P.D, van Heeswijk, W.C, Westerhoff, H.V, Vasudevan, S.G, Ollis, D.L.
登録日1998-07-14
公開日1999-07-23
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献GlnK, a PII-homologue: structure reveals ATP binding site and indicates how the T-loops may be involved in molecular recognition.
J.Mol.Biol., 282, 1998
2OVR
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Structure of the Skp1-Fbw7-CyclinEdegN complex
分子名称: F-box/WD repeat protein 7, S-phase kinase-associated protein 1A, SULFATE ION, ...
著者Hao, B, Oehlmann, S, Sowa, M.E, Harper, J.W, Pavletich, N.P.
登録日2007-02-14
公開日2007-04-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structure of a Fbw7-Skp1-Cyclin E Complex: Multisite-Phosphorylated Substrate Recognition by SCF Ubiquitin Ligases
Mol.Cell, 26, 2007
2GRF
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Crystal structure of Scapharca inaequivalvis HBI, M37V mutant in the absence of ligand
分子名称: Globin-1, PROTOPORPHYRIN IX CONTAINING FE
著者Knapp, J.E, Pahl, R, Srajer, V, Royer Jr, W.E.
登録日2006-04-24
公開日2006-05-09
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Allosteric action in real time: Time-resolved crystallographic studies of a cooperative dimeric hemoglobin.
Proc.Natl.Acad.Sci.Usa, 103, 2006
4LVE
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LEN K30T MUTANT: A DOMAIN FLIP AS A RESULT OF A SINGLE AMINO ACID SUBSTITUTION
分子名称: LEN
著者Schiffer, M, Pokkuluri, P.R.
登録日1998-05-12
公開日1999-05-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献A domain flip as a result of a single amino-acid substitution.
Structure, 6, 1998

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