3GOK
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![BU of 3gok by Molmil](/molmil-images/mine/3gok) | Binding site mapping of protein ligands | 分子名称: | 2-(2-QUINOLIN-3-YLPYRIDIN-4-YL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE, MAP kinase-activated protein kinase 2 | 著者 | Scheich, C. | 登録日 | 2009-03-19 | 公開日 | 2010-03-02 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Binding site mapping of protein ligands To be published
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1WDX
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![BU of 1wdx by Molmil](/molmil-images/mine/1wdx) | Yeast BBC1 SH3 domain, triclinic crystal form | 分子名称: | Myosin tail region-interacting protein MTI1 | 著者 | Wilmanns, M, Consani Textor, L, Kursula, P, Kursula, I, Lehmann, F, Song, Y.H. | 登録日 | 2004-05-19 | 公開日 | 2005-05-31 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of Yeast BBC1 SH3 domain, triclinic crystal form To be Published
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1J41
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![BU of 1j41 by Molmil](/molmil-images/mine/1j41) | Direct observation of photolysis-induced tertiary structural changes in human haemoglobin; Crystal structure of alpha(Ni)-beta(Fe) hemoglobin (laser photolysed) | 分子名称: | BUT-2-ENEDIAL, CARBON MONOXIDE, Hemoglobin alpha Chain, ... | 著者 | Adachi, S, Park, S.-Y, Tame, J.R.H, Shiro, Y, Shibayama, N, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2003-02-21 | 公開日 | 2003-07-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Direct observation of photolysis-induced tertiary structural changes in hemoglobin Proc.Natl.Acad.Sci.USA, 100, 2003
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2QR7
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![BU of 2qr7 by Molmil](/molmil-images/mine/2qr7) | |
1X48
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![BU of 1x48 by Molmil](/molmil-images/mine/1x48) | Solution structure of the second DSRM domain in Interferon-induced, double-stranded RNA-activated protein kinase | 分子名称: | Interferon-induced, double-stranded RNA-activated protein kinase | 著者 | He, F, Muto, Y, Inoue, M, Tarada, T, Shirouzu, M, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-14 | 公開日 | 2005-11-14 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the second DSRM domain in Interferon-induced, double-stranded RNA-activated protein kinase To be Published
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1IR7
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![BU of 1ir7 by Molmil](/molmil-images/mine/1ir7) | |
1IR9
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![BU of 1ir9 by Molmil](/molmil-images/mine/1ir9) | |
1X5H
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![BU of 1x5h by Molmil](/molmil-images/mine/1x5h) | The solution structure of the third fibronectin type III domain of human Neogenin | 分子名称: | Neogenin | 著者 | Tochio, N, Sasagawa, A, Koshiba, S, Inoue, M, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-15 | 公開日 | 2005-11-15 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | The solution structure of the third fibronectin type III domain of human Neogenin To be Published
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1X5X
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![BU of 1x5x by Molmil](/molmil-images/mine/1x5x) | Solution structure of the fibronectin type-III domain of human fibronectin type III domain containing protein 3 | 分子名称: | Fibronectin type-III domain containing protein 3a | 著者 | Yoneyama, M, Tochio, N, Koshiba, S, Inoue, M, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-17 | 公開日 | 2005-11-17 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the fibronectin type-III domain of human fibronectin type III domain containing protein 3 To be Published
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1IP4
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![BU of 1ip4 by Molmil](/molmil-images/mine/1ip4) | G72A HUMAN LYSOZYME | 分子名称: | LYSOZYME C, SODIUM ION | 著者 | Takano, K, Yamagata, Y, Yutani, K. | 登録日 | 2001-04-20 | 公開日 | 2001-11-14 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Role of amino acid residues in left-handed helical conformation for the conformational stability of a protein. Proteins, 45, 2001
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1IRV
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![BU of 1irv by Molmil](/molmil-images/mine/1irv) | |
1WBO
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![BU of 1wbo by Molmil](/molmil-images/mine/1wbo) | fragment based p38 inhibitors | 分子名称: | 2-CHLOROPHENOL, MITOGEN-ACTIVATED PROTEIN KINASE 14 | 著者 | Cleasby, A, Devine, L, Gill, A, Jhoti, H. | 登録日 | 2004-11-04 | 公開日 | 2005-01-27 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Fragment-Based Lead Discovery Using X-Ray Crystallography J.Med.Chem., 48, 2005
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1WBW
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![BU of 1wbw by Molmil](/molmil-images/mine/1wbw) | Identification of novel p38 alpha MAP Kinase inhibitors using fragment-based lead generation. | 分子名称: | 3-(1-NAPHTHYLMETHOXY)PYRIDIN-2-AMINE, MITOGEN-ACTIVATED PROTEIN KINASE 14 | 著者 | Tickle, J, Cleasby, A, Devine, L.A, Jhoti, H. | 登録日 | 2004-11-05 | 公開日 | 2005-11-03 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Identification of Novel P38Alpha Map Kinase Inhibitors Using Fragment-Based Lead Generation J.Med.Chem., 48, 2005
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1IRH
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![BU of 1irh by Molmil](/molmil-images/mine/1irh) | The Solution Structure of The Third Kunitz Domain of Tissue Factor Pathway Inhibitor | 分子名称: | tissue factor pathway inhibitor | 著者 | Mine, S, Yamazaki, T, Miyata, T, Hara, S, Kato, H. | 登録日 | 2001-10-02 | 公開日 | 2002-02-06 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural mechanism for heparin-binding of the third Kunitz domain of human tissue factor pathway inhibitor. Biochemistry, 41, 2002
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1IS0
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![BU of 1is0 by Molmil](/molmil-images/mine/1is0) | Crystal Structure of a Complex of the Src SH2 Domain with Conformationally Constrained Peptide Inhibitor | 分子名称: | AY0 GLU GLU ILE peptide, Tyrosine-protein kinase transforming protein SRC | 著者 | Davidson, J.P, Lubman, O, Rose, T, Waksman, G, Martin, S.F. | 登録日 | 2001-11-02 | 公開日 | 2002-02-06 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Calorimetric and structural studies of 1,2,3-trisubstituted cyclopropanes as conformationally constrained peptide inhibitors of Src SH2 domain binding. J.Am.Chem.Soc., 124, 2002
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2BLP
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![BU of 2blp by Molmil](/molmil-images/mine/2blp) | |
2BLX
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1IWU
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![BU of 1iwu by Molmil](/molmil-images/mine/1iwu) | Crystal Structure Analysis of Human lysozyme at 127K. | 分子名称: | CHLORIDE ION, LYSOZYME C | 著者 | Joti, Y, Nakasako, M, Kidera, A, Go, N. | 登録日 | 2002-06-03 | 公開日 | 2002-09-04 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Nonlinear temperature dependence of the crystal structure of lysozyme: correlation between coordinate shifts and thermal factors. Acta Crystallogr.,Sect.D, 58, 2002
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2XEZ
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![BU of 2xez by Molmil](/molmil-images/mine/2xez) | Crystal structure of checkpoint kinase 1 (Chk1) in complex with inhibitors | 分子名称: | 1,2-ETHANEDIOL, 6-(1H-PYRAZOL-3-YL)-3-(1H-PYRAZOL-4-YL)IMIDAZO[1,2-A]PYRAZINE, SERINE/THREONINE-PROTEIN KINASE CHK1 | 著者 | Matthews, T.P, McHardy, T, Klair, S, Boxall, K, Fisher, M, Cherry, M, Allen, C.E, Addison, G.J, Ellard, J, Aherne, G.W, Westwood, I.M, vanMontfort, R, Garrett, M.D, Reader, J.C, Collins, I. | 登録日 | 2010-05-19 | 公開日 | 2010-07-07 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Design and Evaluation of 3,6-Di(Hetero)Aryl Imidazo[1,2-A]Pyrazines as Inhibitors of Checkpoint and Other Kinases. Bioorg.Med.Chem.Lett., 20, 2010
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2C2C
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![BU of 2c2c by Molmil](/molmil-images/mine/2c2c) | |
1SGC
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![BU of 1sgc by Molmil](/molmil-images/mine/1sgc) | |
1IVC
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![BU of 1ivc by Molmil](/molmil-images/mine/1ivc) | |
1IWX
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![BU of 1iwx by Molmil](/molmil-images/mine/1iwx) | Crystal Structure Analysis of Human lysozyme at 161K. | 分子名称: | CHLORIDE ION, LYSOZYME C | 著者 | Joti, Y, Nakasako, M, Kidera, A, Go, N. | 登録日 | 2002-06-03 | 公開日 | 2002-09-04 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Nonlinear temperature dependence of the crystal structure of lysozyme: correlation between coordinate shifts and thermal factors. Acta Crystallogr.,Sect.D, 58, 2002
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1X3D
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![BU of 1x3d by Molmil](/molmil-images/mine/1x3d) | Solution structure of the fibronectin type-III domain of human fibronectin type-III domain containing protein 3a | 分子名称: | Fibronectin type-III domain containing protein 3a | 著者 | Yoneyama, M, Tochio, N, Koshiba, S, Inoue, M, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-02 | 公開日 | 2005-11-02 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the fibronectin type-III domain of human fibronectin type-III domain containing protein 3a To be Published
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1X4G
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![BU of 1x4g by Molmil](/molmil-images/mine/1x4g) | Solution structure of RRM domain in Nucleolysin TIAR | 分子名称: | Nucleolysin TIAR | 著者 | He, F, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-14 | 公開日 | 2005-11-14 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of RRM domain in Nucleolysin TIAR To be Published
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