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1BQM
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HIV-1 RT/HBY 097
分子名称: (S)-4-ISOPROPOXYCARBONYL-6-METHOXY-3-METHYLTHIOMETHYL-3,4-DIHYDROQUINOXALIN-2(1H)-THIONE, REVERSE TRANSCRIPTASE
著者Hsiou, Y, Das, K, Ding, J, Arnold, E.
登録日1998-08-17
公開日1999-01-06
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structures of Tyr188Leu mutant and wild-type HIV-1 reverse transcriptase complexed with the non-nucleoside inhibitor HBY 097: inhibitor flexibility is a useful design feature for reducing drug resistance.
J.Mol.Biol., 284, 1998
1BQN
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TYR 188 LEU HIV-1 RT/HBY 097
分子名称: (S)-4-ISOPROPOXYCARBONYL-6-METHOXY-3-METHYLTHIOMETHYL-3,4-DIHYDROQUINOXALIN-2(1H)-THIONE, REVERSE TRANSCRIPTASE
著者Hsiou, Y, Das, K, Ding, J, Arnold, E.
登録日1998-08-17
公開日1999-01-06
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structures of Tyr188Leu mutant and wild-type HIV-1 reverse transcriptase complexed with the non-nucleoside inhibitor HBY 097: inhibitor flexibility is a useful design feature for reducing drug resistance.
J.Mol.Biol., 284, 1998
1BQO
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DISCOVERY OF POTENT, ACHIRAL MATRIX METALLOPROTEINASE INHIBITORS
分子名称: 1,3-BIS-(4-METHOXY-BENZENESULFONYL)-5,5-DIMETHYL-HEXAHYDRO-PYRIMIDINE-2-CARBOXYLIC ACID HYDROXYAMIDE, CALCIUM ION, STROMELYSIN-1, ...
著者Pikul, S, Dunham, K.L.M, Almstead, N.G, De, B, Natchus, M.G, Anastasio, M.V, Mcphail, S.J, Snider, C.E, Taiwo, Y.O, Rydel, T.J, Dunaway, C.M, Gu, F, Mieling, G.E.
登録日1998-08-17
公開日1999-08-17
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Discovery of potent, achiral matrix metalloproteinase inhibitors.
J.Med.Chem., 41, 1998
1GFS
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GDP-FUCOSE SYNTHETASE FROM E. COLI
分子名称: GDP-FUCOSE SYNTHETASE
著者Somers, W.S, Stahl, M.L, Sullivan, F.X.
登録日1998-08-17
公開日1999-08-17
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献GDP-fucose synthetase from Escherichia coli: structure of a unique member of the short-chain dehydrogenase/reductase family that catalyzes two distinct reactions at the same active site.
Structure, 6, 1998
3GRX
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BU of 3grx by Molmil
NMR STRUCTURE OF ESCHERICHIA COLI GLUTAREDOXIN 3-GLUTATHIONE MIXED DISULFIDE COMPLEX, 20 STRUCTURES
分子名称: GLUTAREDOXIN 3, GLUTATHIONE
著者Nordstrand, K, Aslund, F, Holmgren, A, Otting, G, Berndt, K.D.
登録日1998-08-17
公開日1999-03-30
最終更新日2018-03-14
実験手法SOLUTION NMR
主引用文献NMR structure of Escherichia coli glutaredoxin 3-glutathione mixed disulfide complex: implications for the enzymatic mechanism.
J.Mol.Biol., 286, 1999
2MYO
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SOLUTION STRUCTURE OF MYOTROPHIN, NMR, MINIMIZED AVERAGE STRUCTURE
分子名称: MYOTROPHIN
著者Yang, Y, Nanduri, S, Sen, S, Qin, J.
登録日1998-08-17
公開日1999-08-17
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献The structural basis of ankyrin-like repeat function as revealed by the solution structure of myotrophin.
Structure, 6, 1998
1MHD
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CRYSTAL STRUCTURE OF A SMAD MH1 DOMAIN BOUND TO DNA
分子名称: DNA, SMAD3
著者Shi, Y.
登録日1998-08-18
公開日1999-08-18
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of a Smad MH1 domain bound to DNA: insights on DNA binding in TGF-beta signaling.
Cell(Cambridge,Mass.), 94, 1998
1BQU
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CYTOKYNE-BINDING REGION OF GP130
分子名称: GLYCEROL, PROTEIN (GP130), SULFATE ION
著者Bravo, J, Staunton, D, Heath, J.K, Jones, E.Y.
登録日1998-08-18
公開日1998-08-26
最終更新日2022-12-21
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of a cytokine-binding region of gp130.
EMBO J., 17, 1998
1BQS
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THE CRYSTAL STRUCTURE OF MUCOSAL ADDRESSIN CELL ADHESION MOLECULE-1 (MADCAM-1)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, PROTEIN (MUCOSAL ADDRESSIN CELL ADHESION MOLECULE-1)
著者Tan, K, Casasnovas, J.M, Liu, J.H, Briskin, M.J, Springer, T.A, Wang, J.-H.
登録日1998-08-18
公開日1999-08-13
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The structure of immunoglobulin superfamily domains 1 and 2 of MAdCAM-1 reveals novel features important for integrin recognition.
Structure, 6, 1998
1BQT
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THREE-DIMENSIONAL STRUCTURE OF HUMAN INSULIN-LIKE GROWTH FACTOR-I (IGF-I) DETERMINED BY 1H-NMR AND DISTANCE GEOMETRY, 6 STRUCTURES
分子名称: INSULIN-LIKE GROWTH FACTOR-I
著者Sato, A, Nishimura, S, Ohkubo, T, Kyogoku, Y, Koyama, S, Kobayashi, M, Yasuda, T, Kobayashi, Y.
登録日1998-08-18
公開日1999-05-18
最終更新日2022-02-16
実験手法SOLUTION NMR
主引用文献Three-dimensional structure of human insulin-like growth factor-I (IGF-I) determined by 1H-NMR and distance geometry.
Int.J.Pept.Protein Res., 41, 1993
1BQQ
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CRYSTAL STRUCTURE OF THE MT1-MMP--TIMP-2 COMPLEX
分子名称: CALCIUM ION, MEMBRANE-TYPE MATRIX METALLOPROTEINASE, METALLOPROTEINASE INHIBITOR 2, ...
著者Fernandez-Catalan, C, Bode, W, Huber, R, Turk, D, Calvete, J.J, Lichte, A, Tschesche, H, Maskos, K.
登録日1998-08-18
公開日1999-08-18
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Crystal structure of the complex formed by the membrane type 1-matrix metalloproteinase with the tissue inhibitor of metalloproteinases-2, the soluble progelatinase A receptor.
EMBO J., 17, 1998
1LDZ
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SOLUTION STRUCTURE OF THE LEAD-DEPENDENT RIBOZYME, NMR, 25 STRUCTURES
分子名称: LEAD-DEPENDENT RIBOZYME
著者Hoogstraten, C.G, Legault, P, Pardi, A.
登録日1998-08-18
公開日1998-11-25
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献NMR solution structure of the lead-dependent ribozyme: evidence for dynamics in RNA catalysis.
J.Mol.Biol., 284, 1998
2LDZ
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SOLUTION STRUCTURE OF THE LEAD-DEPENDENT RIBOZYME, NMR, MINIMIZED AVERAGE STRUCTURE
分子名称: LEAD-DEPENDENT RIBOZYME
著者Hoogstraten, C.G, Legault, P, Pardi, A.
登録日1998-08-18
公開日1999-02-23
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献NMR solution structure of the lead-dependent ribozyme: evidence for dynamics in RNA catalysis.
J.Mol.Biol., 284, 1998
5PGM
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BU of 5pgm by Molmil
SACCHAROMYCES CEREVISIAE PHOSPHOGLYCERATE MUTASE
分子名称: ALANINE, PHOSPHOGLYCERATE MUTASE 1, SULFATE ION
著者Rigden, D.J, Phillips, S.E.V, Fothergill-Gilmore, L.A.
登録日1998-08-19
公開日1999-02-16
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Sulphate ions observed in the 2.12 A structure of a new crystal form of S. cerevisiae phosphoglycerate mutase provide insights into understanding the catalytic mechanism.
J.Mol.Biol., 286, 1999
3BAM
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RESTRICTION ENDONUCLEASE BAMHI COMPLEX WITH DNA AND MANGANESE IONS (POST-REACTIVE COMPLEX)
分子名称: DNA (5'-D(*TP*AP*TP*G)-3'), DNA (5'-D(*TP*AP*TP*GP*GP*AP*TP*CP*CP*AP*TP*A)-3'), DNA (5'-D(P*GP*AP*TP*CP*CP*AP*TP*A)-3'), ...
著者Viadiu, H, Aggarwal, A.K.
登録日1998-08-19
公開日1999-01-13
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The role of metals in catalysis by the restriction endonuclease BamHI.
Nat.Struct.Biol., 5, 1998
2ARG
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FORMATION OF AN AMINO ACID BINDING POCKET THROUGH ADAPTIVE ZIPPERING-UP OF A LARGE DNA HAIRPIN LOOP, NMR, 9 STRUCTURES
分子名称: ARGININEAMIDE, DNA APTAMER [5'-D (*TP*GP*AP*CP*CP*AP*GP*GP*GP*CP*AP*AP*AP*CP*GP*GP*TP*AP* GP*GP*TP*GP*AP*GP*TP*GP*GP*TP*CP*A)-3']
著者Lin, C.H, Wang, W, Jones, R.A, Patel, D.J.
登録日1998-08-19
公開日1999-03-23
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Formation of an amino-acid-binding pocket through adaptive zippering-up of a large DNA hairpin loop.
Chem.Biol., 5, 1998
2BAM
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RESTRICTION ENDONUCLEASE BAMHI COMPLEX WITH DNA AND CALCIUM IONS (PRE-REACTIVE COMPLEX).
分子名称: CALCIUM ION, DNA (5'-D(*TP*AP*TP*GP*GP*AP*TP*CP*CP*AP*TP*A)-3'), PROTEIN (ENDONUCLEASE BAMHI)
著者Viadiu, H, Aggarwal, A.K.
登録日1998-08-19
公開日1999-10-31
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The role of metals in catalysis by the restriction endonuclease BamHI.
Nat.Struct.Biol., 5, 1998
1SKF
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CRYSTAL STRUCTURE OF THE STREPTOMYCES K15 DD-TRANSPEPTIDASE
分子名称: D-ALANYL-D-ALANINE TRANSPEPTIDASE
著者Fonze, E, Charlier, P.
登録日1998-08-20
公開日1999-08-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The crystal structure of a penicilloyl-serine transferase of intermediate penicillin sensitivity. The DD-transpeptidase of streptomyces K15.
J.Biol.Chem., 274, 1999
1MUD
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CATALYTIC DOMAIN OF MUTY FROM ESCHERICHIA COLI, D138N MUTANT COMPLEXED TO ADENINE
分子名称: ADENINE, Adenine DNA glycosylase, GLYCEROL, ...
著者Guan, Y, Tainer, J.A.
登録日1998-08-20
公開日1999-09-20
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献MutY catalytic core, mutant and bound adenine structures define specificity for DNA repair enzyme superfamily.
Nat.Struct.Biol., 5, 1998
1NK1
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NK1 FRAGMENT OF HUMAN HEPATOCYTE GROWTH FACTOR/SCATTER FACTOR (HGF/SF) AT 2.5 ANGSTROM RESOLUTION
分子名称: PROTEIN (HEPATOCYTE GROWTH FACTOR PRECURSOR)
著者Chirgadze, D.Y, Hepple, J.P, Zhou, H, Byrd, R.A, Blundell, T.L, Gherardi, E.
登録日1998-08-20
公開日1999-01-13
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of the NK1 fragment of HGF/SF suggests a novel mode for growth factor dimerization and receptor binding.
Nat.Struct.Biol., 6, 1999
1MUY
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CATALYTIC DOMAIN OF MUTY FROM ESCHERICHIA COLI
分子名称: ADENINE GLYCOSYLASE, GLYCEROL, IMIDAZOLE, ...
著者Guan, Y, Tainer, J.A.
登録日1998-08-20
公開日1999-08-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献MutY catalytic core, mutant and bound adenine structures define specificity for DNA repair enzyme superfamily.
Nat.Struct.Biol., 5, 1998
5PAH
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HUMAN PHENYLALANINE HYDROXYLASE CATALYTIC DOMAIN DIMER WITH BOUND DOPAMINE INHIBITOR
分子名称: FE (III) ION, L-DOPAMINE, PHENYLALANINE 4-MONOOXYGENASE
著者Erlandsen, H, Flatmark, T, Stevens, R.C.
登録日1998-08-20
公開日1999-04-27
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystallographic analysis of the human phenylalanine hydroxylase catalytic domain with bound catechol inhibitors at 2.0 A resolution.
Biochemistry, 37, 1998
1PBI
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CRYSTAL STRUCTURE OF A BOWMAN-BIRK INHIBITOR FROM PEA SEEDS
分子名称: BOWMAN-BIRK PROTEINASE INHIBITOR
著者Li De La Sierra, I, Brunie, S.
登録日1998-08-20
公開日1999-01-27
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Dimeric crystal structure of a Bowman-Birk protease inhibitor from pea seeds.
J.Mol.Biol., 285, 1999
6PAH
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HUMAN PHENYLALANINE HYDROXYLASE CATALYTIC DOMAIN DIMER WITH BOUND L-DOPA (3,4-DIHYDROXYPHENYLALANINE) INHIBITOR
分子名称: 3,4-DIHYDROXYPHENYLALANINE, FE (III) ION, PHENYLALANINE 4-MONOOXYGENASE
著者Erlandsen, H, Flatmark, T, Stevens, R.C.
登録日1998-08-20
公開日1999-04-27
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Crystallographic analysis of the human phenylalanine hydroxylase catalytic domain with bound catechol inhibitors at 2.0 A resolution.
Biochemistry, 37, 1998
1BQ3
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SACCHAROMYCES CEREVISIAE PHOSPHOGLYCERATE MUTASE IN COMPLEX WITH INOSITOL HEXAKISPHOSPHATE
分子名称: INOSITOL HEXAKISPHOSPHATE, PROTEIN (PHOSPHOGLYCERATE MUTASE 1), SULFATE ION
著者Rigden, D.J, Phillips, S.E.V, Fothergill-Gilmore, L.A.
登録日1998-08-20
公開日1998-08-26
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Polyanionic inhibitors of phosphoglycerate mutase: combined structural and biochemical analysis.
J.Mol.Biol., 289, 1999

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