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1I2M
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RAN-RCC1-SO4 COMPLEX
分子名称: GTP-BINDING NUCLEAR PROTEIN RAN, REGULATOR OF CHROMOSOME CONDENSATION 1, SULFATE ION
著者Renault, L, Kuhlmann, J, Henkel, A, Wittinghofer, A.
登録日2001-02-11
公開日2001-05-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.76 Å)
主引用文献Structural basis for guanine nucleotide exchange on Ran by the regulator of chromosome condensation (RCC1).
Cell(Cambridge,Mass.), 105, 2001
1H8M
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Solution structure of ykt6
分子名称: SYNAPTOBREVIN HOMOLOG 1
著者Tochio, H, Tsui, M.M.K, Banfield, D.K, Zhang, M.
登録日2001-02-10
公開日2001-08-07
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献An Autoinhibitory Mechanism for Nonsyntaxin Snare Proteins Revealed by the Structure of Ykt6P
Science, 293, 2001
1HM6
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X-RAY STRUCTURE OF FULL-LENGTH ANNEXIN 1
分子名称: ANNEXIN 1, SULFATE ION
著者Rosengarth, A, Gerke, V, Luecke, H.
登録日2000-12-04
公開日2001-02-28
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献X-ray structure of full-length annexin 1 and implications for membrane aggregation.
J.Mol.Biol., 306, 2001
1F9W
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CRYSTAL STRUCTURES OF MUTANTS REVEAL A SIGNALLING PATHWAY FOR ACTIVATION OF THE KINESIN MOTOR ATPASE
分子名称: ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KAR3, MAGNESIUM ION
著者Yun, M, Zhang, X, Park, C.G, Park, H.W, Endow, S.A.
登録日2000-07-11
公開日2001-06-13
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献A structural pathway for activation of the kinesin motor ATPase.
EMBO J., 20, 2001
1F9T
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CRYSTAL STRUCTURES OF KINESIN MUTANTS REVEAL A SIGNALLING PATHWAY FOR ACTIVATION OF THE MOTOR ATPASE
分子名称: ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KAR3, MAGNESIUM ION
著者Yun, M, Zhang, X, Park, C.-G, Park, H.-W, Endow, S.A.
登録日2000-07-11
公開日2001-06-13
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献A structural pathway for activation of the kinesin motor ATPase.
EMBO J., 20, 2001
1GLJ
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ESCHERICHIA COLI GLYCEROL KINASE MUTANT WITH BOUND ATP ANALOG SHOWING SUBSTANTIAL DOMAIN MOTION
分子名称: GAMMA-ARSONO-BETA, GAMMA-METHYLENEADENOSINE-5'-DIPHOSPHATE, GLYCEROL, ...
著者Bystrom, C.E, Pettigrew, D.W, Branchaud, B.P, Remington, S.J.
登録日1998-09-03
公開日1999-05-18
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal structures of Escherichia coli glycerol kinase variant S58-->W in complex with nonhydrolyzable ATP analogues reveal a putative active conformation of the enzyme as a result of domain motion.
Biochemistry, 38, 1999
1J19
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Crystal structure of the radxin FERM domain complexed with the ICAM-2 cytoplasmic peptide
分子名称: 16-mer peptide from Intercellular adhesion molecule-2, radixin
著者Hamada, K, Shimizu, T, Yonemura, S, Tsukita, S, Tsukita, S, Hakoshima, T.
登録日2002-12-02
公開日2003-03-11
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis of adhesion-molecule recognition by ERM proteins revealed by the crystal structure of the radixin-ICAM-2 complex
EMBO J., 22, 2003
1G2T
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SOLUTION STRUCTURE OF EOTAXIN-3
分子名称: EOTAXIN-3
著者Ye, J, Mayer, K.L, Mayer, M.R, Stone, M.J.
登録日2000-10-20
公開日2002-03-13
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献NMR solution structure and backbone dynamics of the CC chemokine eotaxin-3.
Biochemistry, 40, 2001
1J2J
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Crystal structure of GGA1 GAT N-terminal region in complex with ARF1 GTP form
分子名称: ADP-ribosylation factor 1, ADP-ribosylation factor binding protein GGA1, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Shiba, T, Kawasaki, M, Takatsu, H, Nogi, T, Matsugaki, N, Igarashi, N, Suzuki, M, Kato, R, Nakayama, K, Wakatsuki, S.
登録日2003-01-05
公開日2003-05-06
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Molecular mechanism of membrane recruitment of GGA by ARF in lysosomal protein transport
NAT.STRUCT.BIOL., 10, 2003
1ISN
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Crystal structure of merlin FERM domain
分子名称: merlin
著者Shimizu, T, Seto, A, Maita, N, Hamada, K, Tsukita, S, Tsukita, S, Hakoshima, T.
登録日2001-12-13
公開日2002-04-03
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural basis for neurofibromatosis type 2. Crystal structure of the merlin FERM domain.
J.Biol.Chem., 277, 2002
1IH5
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CRYSTAL STRUCTURE OF AQUAPORIN-1
分子名称: AQUAPORIN-1
著者Ren, G, Reddy, V.S, Cheng, A, Melnyk, P, Mitra, A.K.
登録日2001-04-18
公開日2001-04-25
最終更新日2024-02-07
実験手法ELECTRON CRYSTALLOGRAPHY (3.7 Å)
主引用文献Visualization of a water-selective pore by electron crystallography in vitreous ice.
Proc.Natl.Acad.Sci.USA, 98, 2001
1FQY
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STRUCTURE OF AQUAPORIN-1 AT 3.8 A RESOLUTION BY ELECTRON CRYSTALLOGRAPHY
分子名称: AQUAPORIN-1
著者Murata, K, Mitsuoka, K, Hirai, T, Walz, T, Agre, P, Heymann, J.B, Engel, A, Fujiyoshi, Y.
登録日2000-09-07
公開日2000-10-18
最終更新日2024-04-17
実験手法ELECTRON CRYSTALLOGRAPHY (3.8 Å)
主引用文献Structural determinants of water permeation through aquaporin-1.
Nature, 407, 2000
1GLF
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CRYSTAL STRUCTURES OF ESCHERICHIA COLI GLYCEROL KINASE AND THE MUTANT A65T IN AN INACTIVE TETRAMER: CONFORMATIONAL CHANGES AND IMPLICATIONS FOR ALLOSTERIC REGULATION
分子名称: ADENOSINE-5'-DIPHOSPHATE, GLYCEROL, PHOSPHATE ION, ...
著者Feese, M.D, Faber, H.R, Bystrom, C.E, Pettigrew, D.W, Remington, S.J.
登録日1998-08-30
公開日1998-10-16
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.62 Å)
主引用文献Glycerol kinase from Escherichia coli and an Ala65-->Thr mutant: the crystal structures reveal conformational changes with implications for allosteric regulation.
Structure, 6, 1998
1GLL
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ESCHERICHIA COLI GLYCEROL KINASE MUTANT WITH BOUND ATP ANALOG SHOWING SUBSTANTIAL DOMAIN MOTION
分子名称: GLYCEROL, GLYCEROL KINASE, MAGNESIUM ION, ...
著者Bystrom, C.E, Pettigrew, D.W, Branchaud, B.P, Remington, S.J.
登録日1998-09-24
公開日1999-05-18
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal structures of Escherichia coli glycerol kinase variant S58-->W in complex with nonhydrolyzable ATP analogues reveal a putative active conformation of the enzyme as a result of domain motion.
Biochemistry, 38, 1999
1GML
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crystal structure of the mouse CCT gamma apical domain (triclinic)
分子名称: GLYCEROL, T-COMPLEX PROTEIN 1 SUBUNIT GAMMA
著者Pappenberger, G, Wilsher, J.A, Roe, S.M, Willison, K.R, Pearl, L.H.
登録日2001-09-17
公開日2002-06-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal Structure of the Cct Gamma Apical Domain:: Implications for Substrate Binding to the Eukaryotic Cytosolic Chaperonin
J.Mol.Biol., 318, 2002
1GN1
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crystal structure of the mouse CCT gamma apical domain (monoclinic)
分子名称: CALCIUM ION, CCT-GAMMA
著者Pappenberger, G, Wilsher, J.A, Roe, S.M, Willison, K.R, Pearl, L.H.
登録日2001-10-01
公開日2002-06-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal Structure of the Cct Gamma Apical Domain:: Implications for Substrate Binding to the Eukaryotic Cytosolic Chaperonin
J.Mol.Biol., 318, 2002
1FYN
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PHOSPHOTRANSFERASE
分子名称: 3BP-2, PHOSPHOTRANSFERASE FYN
著者Musacchio, A, Saraste, M, Wilmanns, M.
登録日1995-05-17
公開日1996-11-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献High-resolution crystal structures of tyrosine kinase SH3 domains complexed with proline-rich peptides.
Nat.Struct.Biol., 1, 1994
1JV2
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CRYSTAL STRUCTURE OF THE EXTRACELLULAR SEGMENT OF INTEGRIN ALPHAVBETA3
分子名称: 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Xiong, J.P, Stehle, T, Diefenbach, B, Zhang, R, Dunker, R, Scott, D, Joachimiak, A, Goodman, S.L, Arnaout, M.A.
登録日2001-08-28
公開日2001-10-17
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Crystal structure of the extracellular segment of integrin alpha Vbeta3.
Science, 294, 2001
1IFQ
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Sec22b N-terminal domain
分子名称: GLYCEROL, vesicle trafficking protein Sec22b
著者Gonzalez Jr, L.C, Weis, W.I, Scheller, R.H.
登録日2001-04-13
公開日2001-05-02
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献A novel snare N-terminal domain revealed by the crystal structure of Sec22b.
J.Biol.Chem., 276, 2001
1JX2
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CRYSTAL STRUCTURE OF THE NUCLEOTIDE-FREE DYNAMIN A GTPASE DOMAIN, DETERMINED AS MYOSIN FUSION
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Myosin-2 heavy chain,Dynamin-A, ...
著者Niemann, H.H, Knetsch, M.L.W, Scherer, A, Manstein, D.J, Kull, F.J.
登録日2001-09-05
公開日2001-11-07
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of a dynamin GTPase domain in both nucleotide-free and GDP-bound forms.
EMBO J., 20, 2001
1JEG
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Solution structure of the SH3 domain from C-terminal Src Kinase complexed with a peptide from the tyrosine phosphatase PEP
分子名称: HEMATOPOIETIC CELL PROTEIN-TYROSINE PHOSPHATASE 70Z-PEP, TYROSINE-PROTEIN KINASE CSK
著者Ghose, R, Shekhtman, A, Goger, M.J, Ji, H, Cowburn, D.
登録日2001-06-17
公開日2001-10-31
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献A novel, specific interaction involving the Csk SH3 domain and its natural ligand.
Nat.Struct.Biol., 8, 2001
1JWY
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CRYSTAL STRUCTURE OF THE DYNAMIN A GTPASE DOMAIN COMPLEXED WITH GDP, DETERMINED AS MYOSIN FUSION
分子名称: ADENOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Niemann, H.H, Knetsch, M.L.W, Scherer, A, Manstein, D.J, Kull, F.J.
登録日2001-09-05
公開日2001-11-07
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of a dynamin GTPase domain in both nucleotide-free and GDP-bound forms.
EMBO J., 20, 2001
6EHR
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The crystal structure of the human LAMTOR-RagA CTD-RagC CTD complex
分子名称: Ragulator complex protein LAMTOR1, Ragulator complex protein LAMTOR2, Ragulator complex protein LAMTOR3, ...
著者Scheffzek, K, Naschberger, A.
登録日2017-09-14
公開日2017-10-04
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.898 Å)
主引用文献Crystal structure of the human lysosomal mTORC1 scaffold complex and its impact on signaling.
Science, 358, 2017
7MGJ
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TNNI3K complexed with N-methyl-4-(4-(3-(3-(trifluoromethyl) phenyl) ureido) phenoxy)picolinamide
分子名称: N-methyl-4-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]pyridine-2-carboxamide, Serine/threonine-protein kinase TNNI3K
著者Shewchuk, L.M.
登録日2021-04-12
公開日2021-11-10
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Identification of Diarylurea Inhibitors of the Cardiac-Specific Kinase TNNI3K by Designing Selectivity Against VEGFR2, p38 alpha , and B-Raf.
J.Med.Chem., 64, 2021
7MGK
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TNNI3K complexed with 1-(3,5-dichloro-4-((6-(methylamino)pyrimidin-4-yl)oxy)phenyl)-3-(3-(trifluoromethyl)phenyl)urea
分子名称: N-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-N'-[3-(trifluoromethyl)phenyl]urea, Serine/threonine-protein kinase TNNI3K
著者Shewchuk, L.M.
登録日2021-04-12
公開日2021-11-10
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Identification of Diarylurea Inhibitors of the Cardiac-Specific Kinase TNNI3K by Designing Selectivity Against VEGFR2, p38 alpha , and B-Raf.
J.Med.Chem., 64, 2021

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