4EBL
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4E6X
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![BU of 4e6x by Molmil](/molmil-images/mine/4e6x) | ClbP in complex boron-based inhibitor | 分子名称: | ({[(chloromethyl)sulfonyl]amino}methyl)boronic acid, ClbP peptidase, PHOSPHATE ION | 著者 | Cougnoux, A, Delmas, J, Bonnet, R. | 登録日 | 2012-03-16 | 公開日 | 2013-03-27 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.24 Å) | 主引用文献 | The NRP peptidase ClbP as a target for the inhibition
of genotoxicity, cell proliferation and tumorogenesis
mediated by pks-harboring bacteria To be Published
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4E6W
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4E3O
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4E3N
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4E3M
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![BU of 4e3m by Molmil](/molmil-images/mine/4e3m) | |
4E3L
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4E3K
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4E3J
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4E3I
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4DXC
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4DXB
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4DF6
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![BU of 4df6 by Molmil](/molmil-images/mine/4df6) | |
4DE3
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4DE2
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4DE1
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4DE0
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4DDY
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4DDS
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4D2O
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![BU of 4d2o by Molmil](/molmil-images/mine/4d2o) | Crystal structure of the class A extended-spectrum beta-lactamase PER- 2 | 分子名称: | PER-2 BETA-LACTAMASE | 著者 | Power, P, Herman, R, Ruggiero, M, Kerff, F, Galleni, M, Gutkind, G, Charlier, P, Sauvage, E. | 登録日 | 2014-05-12 | 公開日 | 2014-05-21 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal Structure of the Extended-Spectrum Beta-Lactamase Per- 2 and Insights Into the Role of Specific Residues in the Interaction with Beta-Lactams and Beta-Lactamase Inhibitors. Antimicrob.Agents Chemother., 58, 2014
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4C3Q
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![BU of 4c3q by Molmil](/molmil-images/mine/4c3q) | Neutron structure of a perdeuterated Toho-1 R274N R276N double mutant Beta-lactamase in complex with a fully deuterated boronic acid (BZB) at 100K | 分子名称: | BENZO[B]THIOPHENE-2-BORONIC ACID, BETA-LACTAMASE TOHO-1 | 著者 | Coates, L, Tomanicek, S.J, Schrader, T, Weiss, K.L, Ng, J.D, Ostermann, A. | 登録日 | 2013-08-26 | 公開日 | 2014-07-09 | 最終更新日 | 2017-03-22 | 実験手法 | NEUTRON DIFFRACTION (2.2 Å) | 主引用文献 | Cryogenic Neutron Protein Crystallography: Routine Methods and Potential Benefits J.Appl.Crystallogr., 47, 2014
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4BLM
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4BD1
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![BU of 4bd1 by Molmil](/molmil-images/mine/4bd1) | Neutron structure of a perdeuterated Toho-1 R274N R276N double mutant Beta-lactamase in complex with a fully deuterated boronic acid (BZB) | 分子名称: | BENZO[B]THIOPHENE-2-BORONIC ACID, TOHO-1 BETA-LACTAMASE | 著者 | Tomanicek, S.J, Weiss, K.L, Standaert, R.F, Ostermann, A, Schrader, T.E, Ng, J.D, Coates, L. | 登録日 | 2012-10-04 | 公開日 | 2013-01-16 | 最終更新日 | 2017-03-22 | 実験手法 | NEUTRON DIFFRACTION (2.002 Å) | 主引用文献 | Neutron and X-Ray Crystal Structures of a Perdeuterated Enzyme Inhibitor Complex Reveal the Catalytic Proton Network of the Toho-1 Beta-Lactamase for the Acylation Reaction. J.Biol.Chem., 288, 2013
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4BD0
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![BU of 4bd0 by Molmil](/molmil-images/mine/4bd0) | X-ray structure of a perdeuterated Toho-1 R274N R276N double mutant Beta-lactamase in complex with a fully deuterated boronic acid (BZB) | 分子名称: | BENZO[B]THIOPHENE-2-BORONIC ACID, BETA-LACTAMASE TOHO-1, SULFATE ION | 著者 | Tomanicek, S.J, Weiss, K.L, Standaert, R.F, Ostermann, A, Schrader, T.E, Ng, J.D, Coates, L. | 登録日 | 2012-10-04 | 公開日 | 2013-01-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.207 Å) | 主引用文献 | Neutron and X-Ray Crystal Structures of a Perdeuterated Enzyme Inhibitor Complex Reveal the Catalytic Proton Network of the Toho-1 Beta-Lactamase for the Acylation Reaction. J.Biol.Chem., 288, 2013
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4A5R
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![BU of 4a5r by Molmil](/molmil-images/mine/4a5r) | Crystal structure of class A beta-lactamase from Bacillus licheniformis BS3 with tazobactam | 分子名称: | BETA-LACTAMASE, CARBON DIOXIDE, CITRIC ACID, ... | 著者 | Power, P, Sauvage, E, Herman, R, Kerff, F, Charlier, P. | 登録日 | 2011-10-28 | 公開日 | 2012-10-10 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal Structure of Class a Beta-Lactamase from Bacillus Licheniformis Inhibited by Tazobactam To be Published
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