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6YIO
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CRYSTAL STRUCTURE OF FAB RG6292 IN COMPLEX WITH CD25 ECD
分子名称: FAB FRAGMENT HEAVY CHAIN, FAB FRGAMENT LIGHT CHAIN, Interleukin-2 receptor subunit alpha
著者Benz, J, Koll, H, Leibrock, L.
登録日2020-04-01
公開日2020-11-11
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献CD25-T reg -depleting antibodies preserving IL-2 signaling on effector T cells enhance effector activation and antitumor immunity.
Nat Cancer, 1, 2020
2AWU
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BU of 2awu by Molmil
Synapse associated protein 97 PDZ2 domain variant C378G
分子名称: AHH, Synapse-associated protein 97
著者Von Ossowski, I, Oksanen, E, Von Ossowski, L, Cai, C, Sundberg, M, Goldman, A, Keinanen, K.
登録日2005-09-02
公開日2006-08-29
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献Crystal structure of the second PDZ domain of SAP97 in complex with a GluR-A C-terminal peptide
Febs J., 273, 2006
1QMF
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PENICILLIN-BINDING PROTEIN 2X (PBP-2X) ACYL-ENZYME COMPLEX
分子名称: 2-[CARBOXY-(2-FURAN-2-YL-2-METHOXYIMINO-ACETYLAMINO)-METHYL]-5-METHYL-3,6-DIHYDRO-2H-[1,3]THIAZINE-4-CARBOXYLIC ACID, CEFUROXIME (OCT-3-ENE FORM), PENICILLIN-BINDING PROTEIN 2X
著者Gordon, E.J, Mouz, N, Duee, E, Dideberg, O.
登録日1999-09-28
公開日2000-05-25
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The Crystal Structure of the Penicillin Binding Protein 2X from Streptococcus Pneumoniae and its Acyl-Enzyme Form: Implication in Drug Resistance
J.Mol.Biol., 299, 2000
1ZZ2
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BU of 1zz2 by Molmil
Two Classes of p38alpha MAP Kinase Inhibitors Having a Common Diphenylether Core but Exhibiting Divergent Binding Modes
分子名称: Mitogen-activated protein kinase 14, N-[3-(4-FLUOROPHENOXY)PHENYL]-4-[(2-HYDROXYBENZYL)AMINO]PIPERIDINE-1-SULFONAMIDE, octyl beta-D-glucopyranoside
著者Michelotti, E.L, Moffett, K.K, Springman, E.B, Karpusas, M.
登録日2005-06-13
公開日2005-10-18
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Two classes of p38alpha MAP kinase inhibitors having a common diphenylether core but exhibiting divergent binding modes.
Bioorg.Med.Chem.Lett., 15, 2005
4X6Q
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BU of 4x6q by Molmil
An Isoform-specific Myristylation Switch Targets RIIb PKA Holoenzymes to Membranes
分子名称: cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase type II-beta regulatory subunit
著者Zhang, P, Ye, F, Bastidas, A.C, Kornev, A.P, Ginsberg, M.H, Taylor, S.S.
登録日2014-12-08
公開日2015-07-22
最終更新日2019-12-25
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献An Isoform-Specific Myristylation Switch Targets Type II PKA Holoenzymes to Membranes.
Structure, 23, 2015
5KNZ
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BU of 5knz by Molmil
Human Islet Amyloid Polypeptide Segment 19-SGNNFGAILSS-29 with Early Onset S20G Mutation Determined by MicroED
分子名称: hIAPP(residues 19-29)S20G
著者Krotee, P.A.L, Rodriguez, J.A, Sawaya, M.R, Cascio, D, Shi, D, Nannenga, B.L, Hattne, J, Reyes, F.E, Gonen, T, Eisenberg, D.S.
登録日2016-06-28
公開日2016-12-21
最終更新日2024-03-06
実験手法ELECTRON CRYSTALLOGRAPHY (1.9 Å)
主引用文献Atomic structures of fibrillar segments of hIAPP suggest tightly mated beta-sheets are important for cytotoxicity.
Elife, 6, 2017
7XQM
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BU of 7xqm by Molmil
InDel-mutant short chain Dehydrogenase bound to SAH
分子名称: Dehydrogenase, S-ADENOSYL-L-HOMOCYSTEINE
著者Toledo-Patino, S, Laurino, P.
登録日2022-05-08
公開日2022-12-21
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.71 Å)
主引用文献Insertions and deletions mediated functional divergence of Rossmann fold enzymes.
Proc.Natl.Acad.Sci.USA, 119, 2022
1QFR
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BU of 1qfr by Molmil
NMR SOLUTION STRUCTURE OF PHOSPHOCARRIER PROTEIN HPR FROM ENTEROCOCCUS FAECALIS
分子名称: PHOSPHOCARRIER PROTEIN HPR
著者Maurer, T, Doeker, R, Goerler, A, Hengstenberg, W, Kalbitzer, H.R.
登録日1999-04-13
公開日2001-02-28
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Three-dimensional structure of the histidine-containing phosphocarrier protein (HPr) from Enterococcus faecalis in solution.
Eur.J.Biochem., 268, 2001
2ERL
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BU of 2erl by Molmil
PHEROMONE ER-1 FROM
分子名称: ETHANOL, MATING PHEROMONE ER-1
著者Anderson, D.H, Weiss, M.S, Eisenberg, D.
登録日1995-12-20
公開日1996-07-11
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献A challenging case for protein crystal structure determination: the mating pheromone Er-1 from Euplotes raikovi.
Acta Crystallogr.,Sect.D, 52, 1996
2HIG
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BU of 2hig by Molmil
Crystal Structure of Phosphofructokinase apoenzyme from Trypanosoma brucei.
分子名称: 6-phospho-1-fructokinase, SODIUM ION
著者Martinez-Oyanedel, J, McNae, I.W, Fothergill-Gilmore, L.A, Walkinshaw, M.D.
登録日2006-06-29
公開日2007-02-13
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The First Crystal Structure of Phosphofructokinase from a Eukaryote: Trypanosoma brucei.
J.Mol.Biol., 366, 2007
2A4N
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BU of 2a4n by Molmil
Crystal structure of aminoglycoside 6'-N-acetyltransferase complexed with coenzyme A
分子名称: COENZYME A, SULFATE ION, aac(6')-Ii
著者Burk, D.L, Xiong, B, Breitbach, C, Berghuis, A.M.
登録日2005-06-29
公開日2005-09-20
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structures of aminoglycoside acetyltransferase AAC(6')-Ii in a novel crystal form: structural and normal-mode analyses.
Acta Crystallogr.,Sect.D, 61, 2005
3CAW
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BU of 3caw by Molmil
Crystal structure of o-succinylbenzoate synthase from Bdellovibrio bacteriovorus liganded with Mg
分子名称: MAGNESIUM ION, o-succinylbenzoate synthase
著者Fedorov, A.A, Fedorov, E.V, Sakai, A, Burley, S.K, Gerlt, J.A, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2008-02-20
公開日2008-03-04
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Loss of quaternary structure is associated with rapid sequence divergence in the OSBS family.
Proc.Natl.Acad.Sci.USA, 111, 2014
3CBS
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BU of 3cbs by Molmil
CELLULAR RETINOIC ACID BINDING PROTEIN II IN COMPLEX WITH A SYNTHETIC RETINOIC ACID (RO-12 7310)
分子名称: (2E,4E,6E,8E)-9-(4-hydroxy-2,3,6-trimethylphenyl)-3,7-dimethylnona-2,4,6,8-tetraenoic acid, PROTEIN (CRABP-II)
著者Chaudhuri, B, Kleywegt, G.J, Bergfors, T, Jones, T.A.
登録日1999-02-22
公開日1999-12-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structures of cellular retinoic acid binding proteins I and II in complex with synthetic retinoids.
Acta Crystallogr.,Sect.D, 55, 1999
2FCQ
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X-ray Crystal Structure of a Chemically Synthesized Ubiquitin with a Cubic Space Group
分子名称: CADMIUM ION, Ubiquitin
著者Bang, D, Gribenko, A.V, Tereshko, V, Kossiakoff, A.A, Kent, S.B, Makhatadze, G.I.
登録日2005-12-12
公開日2006-01-31
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Dissecting the energetics of protein alpha-helix C-cap termination through chemical protein synthesis.
Nat.Chem.Biol., 2, 2006
3CBA
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BU of 3cba by Molmil
Crystal structure of Lipopeptide Detergent (LPD-12) (Hexagonal)
分子名称: DECYL-BETA-D-MALTOPYRANOSIDE, LPD-12
著者Ho, D.N, Pomroy, N.C, Cuesta-Seijo, J.A, Prive, G.G.
登録日2008-02-21
公開日2008-09-09
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Packing and Twinning in Orthorhombic and Hexagonal Crystals of Lipopeptide Detergent (LPD-12)
To be Published
1Z3W
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Structure of Phanerochaete chrysosporium cellobiohydrolase Cel7D (CBH58) in complex with cellobioimidazole
分子名称: (5R,6R,7R,8S)-7,8-dihydroxy-5-(hydroxymethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl beta-D-glucopyranoside, 2-acetamido-2-deoxy-beta-D-glucopyranose, cellulase
著者Ubhayasekera, W, Vasella, A, Stahlberg, J, Mowbray, S.L.
登録日2005-03-14
公開日2005-04-26
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structures of Phanerochaete chrysosporium Cel7D in complex with product and inhibitors
Febs J., 272, 2005
1Z3T
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Structure of Phanerochaete chrysosporium cellobiohydrolase Cel7D (CBH58) in complex with cellobiose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose, cellulase
著者Ubhayasekera, W, Stahlberg, J, Mowbray, S.L.
登録日2005-03-14
公開日2005-04-26
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structures of Phanerochaete chrysosporium Cel7D in complex with product and inhibitors
Febs J., 272, 2005
1ML5
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BU of 1ml5 by Molmil
Structure of the E. coli ribosomal termination complex with release factor 2
分子名称: 30S 16S RIBOSOMAL RNA, 30S RIBOSOMAL PROTEIN S10, 30S RIBOSOMAL PROTEIN S11, ...
著者Klaholz, B.P, Pape, T, Zavialov, A.V, Myasnikov, A.G, Orlova, E.V, Vestergaard, B, Ehrenberg, M, van Heel, M.
登録日2002-08-30
公開日2003-01-14
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (14 Å)
主引用文献Structure of the Escherichia coli ribosomal termination complex with release factor 2
Nature, 421, 2003
1Z3V
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Structure of Phanerochaete chrysosporium cellobiohydrolase Cel7D (CBH58) in complex with lactose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, beta-D-galactopyranose-(1-4)-beta-D-glucopyranose, cellulase
著者Ubhayasekera, W, Munoz, I.G, Stahlberg, J, Mowbray, S.L.
登録日2005-03-14
公開日2005-04-26
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Structures of Phanerochaete chrysosporium Cel7D in complex with product and inhibitors
Febs J., 272, 2005
2FCM
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BU of 2fcm by Molmil
X-ray Crystal Structure of a Chemically Synthesized [D-Gln35]Ubiquitin with a Cubic Space Group
分子名称: ACETATE ION, CADMIUM ION, Ubiquitin
著者Bang, D, Gribenko, A.V, Tereshko, V, Kossiakoff, A.A, Kent, S.B, Makhatadze, G.I.
登録日2005-12-12
公開日2006-01-31
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Dissecting the energetics of protein alpha-helix C-cap termination through chemical protein synthesis.
Nat.Chem.Biol., 2, 2006
2JHG
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BU of 2jhg by Molmil
Structural evidence for a ligand coordination switch in liver alcohol dehydrogenase
分子名称: 2-METHYLPROPANAMIDE, ALCOHOL DEHYDROGENASE E CHAIN, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Meijers, R, Adolph, H.W, Dauter, Z, Wilson, K.S, Lamzin, V.S, Cedergren-Zeppezauer, E.S.
登録日2007-02-22
公開日2007-04-24
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Structural Evidence for a Ligand Coordination Switch in Liver Alcohol Dehydrogenase
Biochemistry, 46, 2007
1QME
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PENICILLIN-BINDING PROTEIN 2X (PBP-2X)
分子名称: PENICILLIN-BINDING PROTEIN 2X, SULFATE ION
著者Gordon, E.J, Mouz, N, Duee, E, Dideberg, O.
登録日1999-09-28
公開日2000-05-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The Crystal Structure of the Penicillin-Binding Protein 2X from Streptococcus Pneumoniae and its Acyl-Enzyme Form: Implication in Drug Resistance.
J.Mol.Biol., 299, 2000
3CS9
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BU of 3cs9 by Molmil
Human ABL kinase in complex with nilotinib
分子名称: Nilotinib, Proto-oncogene tyrosine-protein kinase ABL1
著者Cowan-Jacob, S.W, Fendrich, G, Manley, P, Liebetanz, J, Fabbro, D.
登録日2008-04-09
公開日2008-04-22
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.21 Å)
主引用文献Characterization of AMN107, a selective inhibitor of native and mutant Bcr-Abl
Cancer Cell, 7, 2005
1MCV
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Crystal Structure Analysis of a Hybrid Squash Inhibitor in Complex with Porcine Pancreatic Elastase
分子名称: CALCIUM ION, Elastase 1, HEI-TOE I, ...
著者Ay, J, Hilpert, K, Krauss, N, Schneider-Mergener, J, Hoehne, W.
登録日2002-08-06
公開日2003-02-04
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure of a hybrid squash inhibitor in complex with porcine pancreatic elastase at 1.8 A resolution.
Acta Crystallogr.,Sect.D, 59, 2003
1MOU
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Crystal structure of Coral pigment
分子名称: GFP-like non-fluorescent chromoprotein, IODIDE ION
著者Prescott, M, Ling, M, Beddoe, T, Oakley, A.J, Dove, S, Hoegh-Guldberg, O, Devenish, R.J, Rossjohn, J.
登録日2002-09-10
公開日2003-04-08
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The 2.2 a crystal structure of a pocilloporin pigment reveals a nonplanar chromophore conformation.
Structure, 11, 2003

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