8FRD
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8FRC
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8FRB
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8FRA
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8FR9
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8FG7
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8FG5
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![BU of 8fg5 by Molmil](/molmil-images/mine/8fg5) | Apo mouse acidic mammalian chitinase, catalytic domain at 100 K | 分子名称: | Acidic mammalian chitinase, MAGNESIUM ION | 著者 | Diaz, R.E, Correy, G.J, Young, I.D, Thompson, M.C, Fraser, J.S. | 登録日 | 2022-12-12 | 公開日 | 2023-03-01 | 最終更新日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Structural characterization of ligand binding and pH-specific enzymatic activity of mouse Acidic Mammalian Chitinase. Biorxiv, 2024
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8DF1
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![BU of 8df1 by Molmil](/molmil-images/mine/8df1) | Chi3l1 bound by antibody C59 | 分子名称: | C59 Fab Heavy chain, C59 Fab Light chain, Chitinase-3-like protein 1, ... | 著者 | Wrapp, D, McLellan, J.S. | 登録日 | 2022-06-21 | 公開日 | 2023-03-01 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.3 Å) | 主引用文献 | A novel humanized Chi3l1 blocking antibody attenuates acetaminophen-induced liver injury in mice. Antib Ther, 6, 2023
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8C6Z
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![BU of 8c6z by Molmil](/molmil-images/mine/8c6z) | necrotic enteritis associated Clostridium p. chitinase F8UNI4 in complex with inhibitor bisdionin C | 分子名称: | 1,1'-PROPANE-1,3-DIYLBIS(3,7-DIMETHYL-3,7-DIHYDRO-1H-PURINE-2,6-DIONE), CADMIUM ION, COBALT (II) ION, ... | 著者 | Bloch, Y, Savvides, S.N. | 登録日 | 2023-01-12 | 公開日 | 2023-05-31 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Contribution and structural characterization of Chitinases to Clostridium perfringens Pathogenesis in Broilers To Be Published
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7ZYA
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7ZY9
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7Z65
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![BU of 7z65 by Molmil](/molmil-images/mine/7z65) | A GH18 from haloalkaliphilic bacterium unveils environment-dependent variations in the catalytic machinery of chitinases | 分子名称: | 1,2-ETHANEDIOL, Chitinase, GH18 family | 著者 | Madhuprakash, J, Dalhus, B, Rohr, A.K, Bissaro, B, Vaaje-Kolstad, G, Sorlie, M, Eijsink, V.G. | 登録日 | 2022-03-11 | 公開日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.108 Å) | 主引用文献 | A GH18 from haloalkaliphilic bacterium unveils environment-dependent variations in the catalytic machinery of chitinases To Be Published
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7Z64
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![BU of 7z64 by Molmil](/molmil-images/mine/7z64) | A GH18 from haloalkaliphilic bacterium unveils environment-dependent variations in the catalytic machinery of chitinases | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Chitinase, ... | 著者 | Madhuprakash, J, Dalhus, B, Rohr, A.K, Bissaro, B, Vaaje-Kolstad, G, Sorlie, M, Eijsink, V.G. | 登録日 | 2022-03-10 | 公開日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.31 Å) | 主引用文献 | A GH18 from haloalkaliphilic bacterium unveils environment-dependent variations in the catalytic machinery of chitinases To Be Published
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7XMH
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![BU of 7xmh by Molmil](/molmil-images/mine/7xmh) | Crystal structure of a rice class IIIb chitinase, Oschib2 | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, Putative class III chitinase | 著者 | Jun, T, Tomoya, T, Tomoyuki, N, Takayuki, O. | 登録日 | 2022-04-25 | 公開日 | 2023-05-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.18 Å) | 主引用文献 | Characterization of two rice GH18 chitinases belonging to family 8 of plant pathogenesis-related proteins. Plant Sci., 326, 2023
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7VRG
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![BU of 7vrg by Molmil](/molmil-images/mine/7vrg) | Crystal structure of chitinase-h from O. furnacalis in complex with Lynamicin B | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Chitinase, ... | 著者 | Lu, Q, Liu, T, Zhou, Y, Yang, Q. | 登録日 | 2021-10-22 | 公開日 | 2022-03-02 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Lynamicin B is a Potential Pesticide by Acting as a Lepidoptera-Exclusive Chitinase Inhibitor. J.Agric.Food Chem., 69, 2021
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7FD6
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![BU of 7fd6 by Molmil](/molmil-images/mine/7fd6) | Crystal structure of SmChiA in complex with 6a | 分子名称: | 11-methyl-3-(pyridin-3-ylmethyl)-4H-pyrimido[5'',4'':5',6']pyrido[2',3':4,5]pyrimido[1,2-b]pyridine-4,6(3H)-dione, Chitinase A | 著者 | Xi, J, Qing, Y. | 登録日 | 2021-07-16 | 公開日 | 2022-07-20 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Discovery of Conformation Constrained Tetracyclic Compounds as potent Chitinase OfChi-h inhibitor with novel binding mode To Be Published
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7FBT
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![BU of 7fbt by Molmil](/molmil-images/mine/7fbt) | Crystal structure of chitinase (RmChi1) from Rhizomucor miehei (sp p32 2 1, MR) | 分子名称: | Chitinase, MAGNESIUM ION | 著者 | Jiang, Z.Q, Hu, S.Q, Zhu, Q, Liu, Y.C, Ma, J.W, Yan, Q.J, Gao, Y.G, Yang, S.Q. | 登録日 | 2021-07-12 | 公開日 | 2021-08-11 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure of a chitinase (RmChiA) from the thermophilic fungus Rhizomucor miehei with a real active site tunnel. Biochim Biophys Acta Proteins Proteom, 1869, 2021
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7CJ2
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![BU of 7cj2 by Molmil](/molmil-images/mine/7cj2) | Crystal structure of the Fab antibody complexed with human YKL-40 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Chitinase 3-like 1 (Cartilage glycoprotein-39), isoform CRA_a, ... | 著者 | Choi, S, Na, J.H, Lee, S.J, Woo, J.R, Kim, D.Y, Hong, J.T, Lee, W.K. | 登録日 | 2020-07-09 | 公開日 | 2021-07-14 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal structure of the Fab antibody complexed with human YKL-40 To Be Published
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7CB1
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![BU of 7cb1 by Molmil](/molmil-images/mine/7cb1) | Structure of Serratia marcescens chitinase B complexed with compound 6q | 分子名称: | 6-azanyl-11-methyl-2-oxidanylidene-N-[(1S)-1-pyridin-3-ylethyl]-1,7,9-triazatricyclo[8.4.0.0^{3,8}]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide, Chitinase B | 著者 | Jiang, X, Yuan, P.T. | 登録日 | 2020-06-10 | 公開日 | 2021-06-16 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Discovery of novel Chitinase Inhibitors with a scaffold of dipyridopyrimidine-3-carboxamide via Structure-based Rational Design To Be Published
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7C92
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![BU of 7c92 by Molmil](/molmil-images/mine/7c92) | Structure of Serratia marcescens chitinase B complexed with compound 6k | 分子名称: | 6-azanyl-11-methyl-2-oxidanylidene-N-(pyridin-3-ylmethyl)-1,7,9-triazatricyclo[8.4.0.0^3,8]tetradeca-3(8),4,6,9,11,13-hexaene-5-carboxamide, Chitinase | 著者 | Jiang, X, Yuan, P.T. | 登録日 | 2020-06-04 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.32 Å) | 主引用文献 | Discovery of novel Chitinase Inhibitors with a scaffold of dipyridopyrimidine-3-carboxamide via Structure-based Rational Design To Be Published
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7C34
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7AKQ
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6ZE8
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![BU of 6ze8 by Molmil](/molmil-images/mine/6ze8) | Crystal structure of human chitotriosidase-1 (hCHIT) catalytic domain in complex with compound OATD-01 | 分子名称: | 5-(4-((2S,5S)-5-(4-chlorobenzyl)-2-methylmorpholino)piperidin-1-yl)-4H-1,2,4-triazol-3-amine, Chitotriosidase-1, GLYCEROL, ... | 著者 | Nowotny, M, Bartlomiejczak, A, Napiorkowska-Gromadzka, A. | 登録日 | 2020-06-16 | 公開日 | 2020-11-11 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Discovery of OATD-01 , a First-in-Class Chitinase Inhibitor as Potential New Therapeutics for Idiopathic Pulmonary Fibrosis. J.Med.Chem., 63, 2020
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6YN4
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6YLJ
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