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1HVR
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RATIONAL DESIGN OF POTENT, BIOAVAILABLE, NONPEPTIDE CYCLIC UREAS AS HIV PROTEASE INHIBITORS
分子名称: HIV-1 PROTEASE, [4R-(4ALPHA,5ALPHA,6BETA,7BETA)]-HEXAHYDRO-5,6-DIHYDROXY-1,3-BIS[2-NAPHTHYL-METHYL]-4,7-BIS(PHENYLMETHYL)-2H-1,3-DIAZEPIN-2-ONE
著者Chang, C.-H.
登録日1994-02-14
公開日1995-01-26
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Rational design of potent, bioavailable, nonpeptide cyclic ureas as HIV protease inhibitors.
Science, 263, 1994
1IDB
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BU of 1idb by Molmil
Crystal structures of HIV-2 protease in complex with inhibitors containing the hydroxyethylamine dipeptide isostere
分子名称: (2R,4S)-N-tert-butyl-1-[(2S,3S)-3-{[(2,6-dimethylphenoxy)acetyl]amino}-2-hydroxy-4-phenylbutyl]-4-(pyridin-4-ylsulfonyl)piperidine-2-carboxamide, Protease
著者Tong, L, Anderson, P.C.
登録日1994-10-19
公開日1995-01-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structures of HIV-2 protease in complex with inhibitors containing the hydroxyethylamine dipeptide isostere.
Structure, 3, 1995
1ETA
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BU of 1eta by Molmil
THE X-RAY CRYSTAL STRUCTURE REFINEMENTS OF NORMAL HUMAN TRANSTHYRETIN AND THE AMYLOIDOGENIC VAL 30-->MET VARIANT TO 1.7 ANGSTROMS RESOLUTION
分子名称: 3,5,3',5'-TETRAIODO-L-THYRONINE, TRANSTHYRETIN
著者Braden, B.C, Steinrauf, L.K, Hamilton, J.A.
登録日1993-05-12
公開日1995-01-26
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The x-ray crystal structure refinements of normal human transthyretin and the amyloidogenic Val-30-->Met variant to 1.7-A resolution.
J.Biol.Chem., 268, 1993
1AMC
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BU of 1amc by Molmil
SOLUTION STRUCTURE OF RESIDUES 1-28 OF THE AMYLOID BETA-PEPTIDE
分子名称: AMYLOID BETA-PEPTIDE
著者Talafous, J, Marcinowski, K.J, Klopman, G, Zagorski, M.G.
登録日1994-11-14
公開日1995-01-26
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of residues 1-28 of the amyloid beta-peptide.
Biochemistry, 33, 1994
1OLG
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BU of 1olg by Molmil
HIGH-RESOLUTION SOLUTION STRUCTURE OF THE OLIGOMERIZATION DOMAIN OF P53 BY MULTI-DIMENSIONAL NMR
分子名称: TUMOR SUPPRESSOR P53 (OLIGOMERIZATION DOMAIN)
著者Clore, G.M, Omichinski, J.G, Gronenborn, A.M.
登録日1994-06-13
公開日1995-01-26
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献High-resolution structure of the oligomerization domain of p53 by multidimensional NMR.
Science, 265, 1994
1ETB
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BU of 1etb by Molmil
THE X-RAY CRYSTAL STRUCTURE REFINEMENTS OF NORMAL HUMAN TRANSTHYRETIN AND THE AMYLOIDOGENIC VAL 30-->MET VARIANT TO 1.7 ANGSTROMS RESOLUTION
分子名称: 3,5,3',5'-TETRAIODO-L-THYRONINE, TRANSTHYRETIN
著者Braden, B.C, Steinrauf, L.K, Hamilton, J.A.
登録日1993-05-12
公開日1995-01-26
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The x-ray crystal structure refinements of normal human transthyretin and the amyloidogenic Val-30-->Met variant to 1.7-A resolution.
J.Biol.Chem., 268, 1993
1INP
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BU of 1inp by Molmil
CRYSTAL STRUCTURE OF INOSITOL POLYPHOSPHATE 1-PHOSPHATASE AT 2.3 ANGSTROMS RESOLUTION
分子名称: INOSITOL POLYPHOSPHATE 1-PHOSPHATASE, MAGNESIUM ION
著者York, J.D, Ponder, J.W, Chen, Z, Mathews, F.S, Majerus, P.W.
登録日1994-10-04
公開日1995-01-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of inositol polyphosphate 1-phosphatase at 2.3-A resolution.
Biochemistry, 33, 1994
2HHD
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OXYGEN AFFINITY MODULATION BY THE N-TERMINI OF THE BETA-CHAINS IN HUMAN AND BOVINE HEMOGLOBIN
分子名称: HEMOGLOBIN (DEOXY) (ALPHA CHAIN), HEMOGLOBIN (DEOXY) (BETA CHAIN), PROTOPORPHYRIN IX CONTAINING FE, ...
著者Gilliland, G.L, Pechik, I, Fronticelli, C, Ji, X.
登録日1994-09-29
公開日1995-01-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystallographic, molecular modeling, and biophysical characterization of the valine beta 67 (E11)-->threonine variant of hemoglobin.
Biochemistry, 35, 1996
2HHE
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BU of 2hhe by Molmil
OXYGEN AFFINITY MODULATION BY THE N-TERMINI OF THE BETA CHAINS IN HUMAN AND BOVINE HEMOGLOBIN
分子名称: HEMOGLOBIN (DEOXY) (ALPHA CHAIN), HEMOGLOBIN (DEOXY) (BETA CHAIN), PROTOPORPHYRIN IX CONTAINING FE
著者Gilliland, G.L, Pechik, I, Fronticelli, C, Ji, X.
登録日1994-09-29
公開日1995-01-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Chloride ion independence of the Bohr effect in a mutant human hemoglobin beta (V1M+H2deleted).
J.Biol.Chem., 269, 1994
1NTR
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BU of 1ntr by Molmil
SOLUTION STRUCTURE OF THE N-TERMINAL RECEIVER DOMAIN OF NTRC
分子名称: NTRC RECEIVER DOMAIN
著者Volkman, B.F, Nohaile, M.J, Amy, N.K, Kustu, S, Wemmer, D.E.
登録日1994-09-16
公開日1995-01-26
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Three-dimensional solution structure of the N-terminal receiver domain of NTRC.
Biochemistry, 34, 1995
1HRM
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BU of 1hrm by Molmil
THE PROXIMAL LIGAND VARIANT HIS93TYR OF HORSE HEART MYOGLOBIN
分子名称: MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION
著者Burk, D.L, Brayer, G.D.
登録日1994-09-21
公開日1995-01-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The proximal ligand variant His93Tyr of horse heart myoglobin.
Biochemistry, 34, 1995
1SCY
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BU of 1scy by Molmil
DETERMINATION OF THE THREE-DIMENSIONAL STRUCTURE OF SCYLLATOXIN BY 1H NUCLEAR MAGNETIC RESONANCE
分子名称: SCYLLATOXIN
著者Martins, J.C, Van De Ven, F.J.M, Borremans, F.A.M.
登録日1994-06-02
公開日1995-01-26
最終更新日2017-11-29
実験手法SOLUTION NMR
主引用文献Determination of the three-dimensional solution structure of scyllatoxin by 1H nuclear magnetic resonance.
J.Mol.Biol., 253, 1995
1BTL
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BU of 1btl by Molmil
CRYSTAL STRUCTURE OF ESCHERICHIA COLI TEM1 BETA-LACTAMASE AT 1.8 ANGSTROMS RESOLUTION
分子名称: BETA-LACTAMASE TEM1, SULFATE ION
著者Jelsch, C, Mourey, L, Masson, J.M, Samama, J.P.
登録日1993-11-01
公開日1995-01-26
最終更新日2019-08-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of Escherichia coli TEM1 beta-lactamase at 1.8 A resolution.
Proteins, 16, 1993
1SLA
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BU of 1sla by Molmil
X-RAY CRYSTALLOGRAPHY REVEALS CROSSLINKING OF MAMMALIAN LECTIN (GALECTIN-1) BY BIANTENNARY COMPLEX TYPE SACCHARIDES
分子名称: BOVINE GALECTIN-1, beta-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[beta-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose
著者Bourne, Y, Cambillau, C.
登録日1994-03-12
公開日1995-01-26
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Crosslinking of mammalian lectin (galectin-1) by complex biantennary saccharides.
Nat.Struct.Biol., 1, 1994
1RMN
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BU of 1rmn by Molmil
A THREE-DIMENSIONAL MODEL FOR THE HAMMERHEAD RIBOZYME BASED ON FLUORESCENCE MEASUREMENTS
分子名称: RNA (49-MER)
著者Tuschl, T, Gohlke, C, Jovin, T.M, Westhof, E, Eckstein, F.
登録日1994-10-20
公開日1995-01-26
最終更新日2024-02-14
実験手法FLUORESCENCE TRANSFER
主引用文献A three-dimensional model for the hammerhead ribozyme based on fluorescence measurements.
Science, 266, 1994
1RCF
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BU of 1rcf by Molmil
STRUCTURE OF THE TRIGONAL FORM OF RECOMBINANT OXIDIZED FLAVODOXIN FROM ANABAENA 7120 AT 1.40 ANGSTROMS RESOLUTION
分子名称: FLAVIN MONONUCLEOTIDE, FLAVODOXIN, SULFATE ION
著者Burkhart, B, Ramakrishnan, B, Yan, H, Reedstrom, R, Markley, J, Straus, N, Sundaralingam, M.
登録日1994-10-31
公開日1995-01-26
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structure of the trigonal form of recombinant oxidized flavodoxin from Anabaena 7120 at 1.40 A resolution.
Acta Crystallogr.,Sect.D, 51, 1995
1RPL
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BU of 1rpl by Molmil
2.3 ANGSTROMS CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF DNA POLYMERASE BETA
分子名称: DNA POLYMERASE BETA
著者Davies II, J.F, Almassy, R.J.
登録日1994-10-25
公開日1995-01-26
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献2.3 A crystal structure of the catalytic domain of DNA polymerase beta.
Cell(Cambridge,Mass.), 76, 1994
2EBN
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BU of 2ebn by Molmil
CRYSTAL STRUCTURE OF ENDO-BETA-N-ACETYLGLUCOSAMINIDASE F1, AN ALPHA(SLASH)BETA-BARREL ENZYME ADAPTED FOR A COMPLEX SUBSTRATE
分子名称: ENDO-BETA-N-ACETYLGLUCOSAMINIDASE F1, ZINC ION
著者Van Roey, P.
登録日1994-08-30
公開日1995-01-26
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of endo-beta-N-acetylglucosaminidase F1, an alpha/beta-barrel enzyme adapted for a complex substrate.
Biochemistry, 33, 1994
1CSV
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REPLACEMENTS IN A CONSERVED LEUCINE CLUSTER IN THE HYDROPHOBIC HEME POCKET OF CYTOCHROME C
分子名称: CYTOCHROME C, HEME C, SULFATE ION
著者Lo, T.P, Brayer, G.D.
登録日1994-10-04
公開日1995-01-26
最終更新日2021-03-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Replacements in a conserved leucine cluster in the hydrophobic heme pocket of cytochrome c.
Protein Sci., 4, 1995
1CSX
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BU of 1csx by Molmil
REPLACEMENTS IN A CONSERVED LEUCINE CLUSTER IN THE HYDROPHOBIC HEME POCKET OF CYTOCHROME C
分子名称: CYTOCHROME C, HEME C, SULFATE ION
著者Lo, T.P, Brayer, G.D.
登録日1994-10-04
公開日1995-01-26
最終更新日2021-03-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Replacements in a conserved leucine cluster in the hydrophobic heme pocket of cytochrome c.
Protein Sci., 4, 1995
1CSU
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BU of 1csu by Molmil
REPLACEMENTS IN A CONSERVED LEUCINE CLUSTER IN THE HYDROPHOBIC HEME POCKET OF CYTOCHROME C
分子名称: CYTOCHROME C, HEME C, SULFATE ION
著者Lo, T.P, Brayer, G.D.
登録日1994-10-04
公開日1995-01-26
最終更新日2021-03-10
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Replacements in a conserved leucine cluster in the hydrophobic heme pocket of cytochrome c.
Protein Sci., 4, 1995
1CSW
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BU of 1csw by Molmil
REPLACEMENTS IN A CONSERVED LEUCINE CLUSTER IN THE HYDROPHOBIC HEME POCKET OF CYTOCHROME C
分子名称: CYTOCHROME C, HEME C, SULFATE ION
著者Lo, T.P, Brayer, G.D.
登録日1994-10-04
公開日1995-01-26
最終更新日2021-03-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Replacements in a conserved leucine cluster in the hydrophobic heme pocket of cytochrome c.
Protein Sci., 4, 1995
1CIH
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BU of 1cih by Molmil
STRUCTURAL AND FUNCTIONAL EFFECTS OF MULTIPLE MUTATIONS AT DISTAL SITES IN CYTOCHROME C
分子名称: CYTOCHROME C, HEME C, SULFATE ION
著者Lo, T.P, Brayer, G.D.
登録日1994-09-26
公開日1995-01-26
最終更新日2021-03-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural and functional effects of multiple mutations at distal sites in cytochrome c.
Biochemistry, 34, 1995
1IDA
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BU of 1ida by Molmil
CRYSTAL STRUCTURES OF HIV-2 PROTEASE IN COMPLEX WITH INHIBITORS CONTAINING THE HYDROXYETHYLAMINE DIPEPTIDE ISOSTERE
分子名称: N-[(1R)-1-{[(1S,2S)-1-benzyl-3-{(2R,4S)-2-(tert-butylcarbamoyl)-4-[(pyridin-3-ylmethyl)sulfanyl]piperidin-1-yl}-2-hydroxypropyl]carbamoyl}-2-methylpropyl]quinoline-2-carboxamide, Protease
著者Tong, L, Anderson, P.C.
登録日1994-10-19
公開日1995-01-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of HIV-2 protease in complex with inhibitors containing the hydroxyethylamine dipeptide isostere.
Structure, 3, 1995
153L
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THE REFINED STRUCTURES OF GOOSE LYSOZYME AND ITS COMPLEX WITH A BOUND TRISACCHARIDE SHOW THAT THE "GOOSE-TYPE LYSOZYMES LACK A CATALYTIC ASPARTATE
分子名称: GOOSE LYSOZYME
著者Weaver, L.H, Gruetter, M.G, Matthews, B.W.
登録日1994-05-05
公開日1995-01-26
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献The refined structures of goose lysozyme and its complex with a bound trisaccharide show that the "goose-type" lysozymes lack a catalytic aspartate residue.
J.Mol.Biol., 245, 1995

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