PDB クエリの検索結果 - 日本蛋白質構造データバンク

PDB: 2 件

Crystal structure of the human HIPK3 kinase domain
分子名称:	1,2-ETHANEDIOL, Homeodomain-interacting protein kinase 3
著者	Kaltheuner, I.H, Anand, K, Geyer, M.
登録日	2021-04-13
公開日	2021-11-24
最終更新日	2024-01-31
実験手法	X-RAY DIFFRACTION (2.5 Å)
主引用文献	Abemaciclib is a potent inhibitor of DYRK1A and HIP kinases involved in transcriptional regulation. Nat Commun, 12, 2021

Crystal structure of the human HIPK3 kinase domain bound to abemaciclib
分子名称:	Homeodomain-interacting protein kinase 3, N-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1H-benzimidazol-6-yl]py rimidin-2-amine
著者	Kaltheuner, I.H, Anand, K, Geyer, M.
登録日	2021-04-13
公開日	2021-11-24
最終更新日	2024-05-01
実験手法	X-RAY DIFFRACTION (2.81 Å)
主引用文献	Abemaciclib is a potent inhibitor of DYRK1A and HIP kinases involved in transcriptional regulation. Nat Commun, 12, 2021