8AAK
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![BU of 8aak by Molmil](/molmil-images/mine/8aak) | Crystal structure of the PDZ tandem of syntenin in complex with compound 29 | 分子名称: | (2~{S})-2-[[(2~{S})-2-(3-oxidanylidene-1~{H}-isoindol-2-yl)-3-phenyl-propanoyl]amino]propanoic acid, GLYCEROL, Syntenin-1 | 著者 | Feracci, M, Barral, K. | 登録日 | 2022-07-01 | 公開日 | 2023-04-26 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.554 Å) | 主引用文献 | Discovery of a PDZ Domain Inhibitor Targeting the Syndecan/Syntenin Protein-Protein Interaction: A Semi-Automated "Hit Identification-to-Optimization" Approach. J.Med.Chem., 66, 2023
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8AAP
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![BU of 8aap by Molmil](/molmil-images/mine/8aap) | Crystal structure of the PDZ tandem of syntenin in complex with compound SYNTi | 分子名称: | (2S)-2-[[(2S)-2-(6-bromanyl-3-oxidanylidene-1H-isoindol-2-yl)-3-[4-(5-ethanoyl-2-fluoranyl-phenyl)phenyl]propanoyl]amino]propanoic acid, Syntenin-1 | 著者 | Feracci, M, Barral, K. | 登録日 | 2022-07-01 | 公開日 | 2023-04-26 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.174 Å) | 主引用文献 | Discovery of a PDZ Domain Inhibitor Targeting the Syndecan/Syntenin Protein-Protein Interaction: A Semi-Automated "Hit Identification-to-Optimization" Approach. J.Med.Chem., 66, 2023
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8AAO
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![BU of 8aao by Molmil](/molmil-images/mine/8aao) | Crystal structure of the PDZ tandem of syntenin in complex with compound 95 | 分子名称: | (2~{S})-2-[[(2~{S})-3-[4-(5-ethanoyl-2-fluoranyl-phenyl)phenyl]-2-(3-oxidanylidene-1~{H}-isoindol-2-yl)propanoyl]amino]propanoic acid, Syntenin-1 | 著者 | Feracci, M, Barral, K. | 登録日 | 2022-07-01 | 公開日 | 2023-04-26 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.469 Å) | 主引用文献 | Discovery of a PDZ Domain Inhibitor Targeting the Syndecan/Syntenin Protein-Protein Interaction: A Semi-Automated "Hit Identification-to-Optimization" Approach. J.Med.Chem., 66, 2023
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8AAI
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1GQ4
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![BU of 1gq4 by Molmil](/molmil-images/mine/1gq4) | |
5VWK
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![BU of 5vwk by Molmil](/molmil-images/mine/5vwk) | |
5VWI
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![BU of 5vwi by Molmil](/molmil-images/mine/5vwi) | |
1GQ5
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![BU of 1gq5 by Molmil](/molmil-images/mine/1gq5) | |
1I16
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![BU of 1i16 by Molmil](/molmil-images/mine/1i16) | STRUCTURE OF INTERLEUKIN 16: IMPLICATIONS FOR FUNCTION, NMR, 20 STRUCTURES | 分子名称: | INTERLEUKIN 16 | 著者 | Muehlhahn, P, Zweckstetter, M, Georgescu, J, Ciosto, C, Renner, C, Lanzendoerfer, M, Lang, K, Ambrosius, D, Baier, M, Kurth, R, Holak, T.A. | 登録日 | 1998-05-20 | 公開日 | 1999-05-25 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure of interleukin 16 resembles a PDZ domain with an occluded peptide binding site. Nat.Struct.Biol., 5, 1998
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4G69
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1I92
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![BU of 1i92 by Molmil](/molmil-images/mine/1i92) | |
4E35
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5WOU
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4F8K
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![BU of 4f8k by Molmil](/molmil-images/mine/4f8k) | Molecular analysis of the interaction between the prostacyclin receptor and the first PDZ domain of PDZK1 | 分子名称: | Na(+)/H(+) exchange regulatory cofactor NHE-RF3, Prostacyclin receptor | 著者 | Kocher, O, Birrane, G, Kinsella, B.T, Mulvaney, E.P. | 登録日 | 2012-05-17 | 公開日 | 2013-02-27 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Molecular Analysis of the Prostacyclin Receptor's Interaction with the PDZ1 Domain of Its Adaptor Protein PDZK1. Plos One, 8, 2013
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4H11
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![BU of 4h11 by Molmil](/molmil-images/mine/4h11) | Interaction partners of PSD-93 studied by X-ray crystallography and fluorescent polarization spectroscopy | 分子名称: | ACETATE ION, Disks large homolog 2, SULFATE ION | 著者 | Fiorentini, M, Kastrup, J.S, Gajhede, M. | 登録日 | 2012-09-10 | 公開日 | 2013-04-03 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Interaction partners of PSD-93 studied by X-ray crystallography and fluorescence polarization spectroscopy. Acta Crystallogr.,Sect.D, 69, 2013
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1IU2
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![BU of 1iu2 by Molmil](/molmil-images/mine/1iu2) | The first PDZ domain of PSD-95 | 分子名称: | PSD-95 | 著者 | Long, J.-F, Tochio, H, Wang, P, Sala, C, Niethammer, M, Sheng, M, Zhang, M. | 登録日 | 2002-02-19 | 公開日 | 2003-03-11 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Supramodular structure and synergistic target binding of the N-terminal tandem PDZ domains of PSD-95 J.MOL.BIOL., 327, 2003
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4GVD
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![BU of 4gvd by Molmil](/molmil-images/mine/4gvd) | Crystal Structure of T-cell Lymphoma Invasion and Metastasis-1 PDZ in complex with Syndecan1 Peptide | 分子名称: | 5-(DIMETHYLAMINO)-1-NAPHTHALENESULFONIC ACID(DANSYL ACID), CHLORIDE ION, SODIUM ION, ... | 著者 | Liu, X, Shepherd, T.R, Murray, A.M, Xu, Z, Fuentes, E.J. | 登録日 | 2012-08-30 | 公開日 | 2013-03-13 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | The structure of the Tiam1 PDZ domain/ phospho-syndecan1 complex reveals a ligand conformation that modulates protein dynamics. Structure, 21, 2013
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1IHJ
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5V6B
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![BU of 5v6b by Molmil](/molmil-images/mine/5v6b) | Crystal structure of GIPC1 | 分子名称: | PDZ domain-containing protein GIPC1 | 著者 | Shang, G, Zhang, X. | 登録日 | 2017-03-16 | 公開日 | 2017-05-31 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure analyses reveal a regulated oligomerization mechanism of the PlexinD1/GIPC/myosin VI complex. Elife, 6, 2017
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5VWC
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5W72
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4GVC
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![BU of 4gvc by Molmil](/molmil-images/mine/4gvc) | Crystal Structure of T-cell Lymphoma Invasion and Metastasis-1 PDZ in complex with phosphorylated Syndecan1 Peptide | 分子名称: | 5-(DIMETHYLAMINO)-1-NAPHTHALENESULFONIC ACID(DANSYL ACID), CHLORIDE ION, SODIUM ION, ... | 著者 | Liu, X, Shepherd, T.R, Murray, A.M, Xu, Z, Fuentes, E.J. | 登録日 | 2012-08-30 | 公開日 | 2013-03-13 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | The structure of the Tiam1 PDZ domain/ phospho-syndecan1 complex reveals a ligand conformation that modulates protein dynamics. Structure, 21, 2013
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4HOP
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![BU of 4hop by Molmil](/molmil-images/mine/4hop) | Crystal structure of the computationally designed NNOS-Syntrophin complex | 分子名称: | Alpha-1-syntrophin, Nitric oxide synthase, brain | 著者 | Harwood, I.M, Melero, C, Ollikainen, N, Kortemme, T. | 登録日 | 2012-10-22 | 公開日 | 2013-11-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.29 Å) | 主引用文献 | Quantification of the transferability of a designed protein specificity switch reveals extensive epistasis in molecular recognition. Proc.Natl.Acad.Sci.USA, 111, 2014
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1GM1
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![BU of 1gm1 by Molmil](/molmil-images/mine/1gm1) | Second PDZ Domain (PDZ2) of PTP-BL | 分子名称: | PROTEIN TYROSINE PHOSPHATASE | 著者 | Walma, T, Tessari, M, Aelen, J, Schepens, J, Hendriks, W, Vuister, G.W. | 登録日 | 2001-09-06 | 公開日 | 2002-03-08 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure, dynamics and binding characteristics of the second PDZ domain of PTP-BL. J. Mol. Biol., 316, 2002
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1IU0
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![BU of 1iu0 by Molmil](/molmil-images/mine/1iu0) | The first PDZ domain of PSD-95 | 分子名称: | PSD-95 | 著者 | Long, J.-F, Tochio, H, Wang, P, Sala, C, Niethammer, M, Sheng, M, Zhang, M. | 登録日 | 2002-02-18 | 公開日 | 2003-03-11 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Supramodular structure and synergistic target binding of the N-terminal tandem PDZ domains of PSD-95 J.MOL.BIOL., 327, 2003
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