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PDB: 73 件

6GY5
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BU of 6gy5 by Molmil
Crystal structure of the kelch domain of human KLHL20 in complex with DAPK1 peptide
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Death-associated protein kinase 1, ...
著者Chen, Z, Hozjan, V, Strain-Damerell, C, Williams, E, Wang, D, Cooper, C.D.O, Sanvitale, C.E, Fairhead, M, Carpenter, E.P, Pike, A.C.W, Krojer, T, Srikannathasan, V, Sorrell, F, Johansson, C, Mathea, S, Burgess-Brown, N, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Bullock, A.N.
登録日2018-06-28
公開日2018-08-08
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.086 Å)
主引用文献Structural Basis for Recruitment of DAPK1 to the KLHL20 E3 Ligase.
Structure, 27, 2019
4PF4
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BU of 4pf4 by Molmil
1.1A X-RAY STRUCTURE OF THE APO CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE 1, aa 1-277
分子名称: Death-associated protein kinase 1, GLYCEROL, MAGNESIUM ION, ...
著者Temmerman, K, Simon, B, Wilmanns, M.
登録日2014-04-28
公開日2014-05-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.13 Å)
主引用文献1.1A X-RAY STRUCTURE OF THE APO CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE 1, aa 1-277
To Be Published
2W4J
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BU of 2w4j by Molmil
X-ray structure of a DAP-Kinase 2-277
分子名称: ACETATE ION, ADENOSINE-5'-DIPHOSPHATE, DEATH-ASSOCIATED PROTEIN KINASE 1, ...
著者De Diego, I, Kuper, J, Lehmann, F, Wilmanns, M.
登録日2008-11-27
公開日2009-12-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献X-Ray Structure of a Dap-Kinase Calmodulin Complex
To be Published
3GU4
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BU of 3gu4 by Molmil
Crystal structure of DAPKQ23V-AMPPNP
分子名称: Death-associated protein kinase 1, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者McNamara, L.K, Schavocky, J.S, Watterson, D.M, Brunzelle, J.S.
登録日2009-03-28
公開日2010-03-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Enzymatic activity and crystallgoraphic analyses of a glycine-rich loop mutant of DAPK
To be Published
7CCW
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BU of 7ccw by Molmil
Crystal structure of death-associated protein kinase 1 in complex with resveratrol and MES
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Death-associated protein kinase 1, RESVERATROL, ...
著者Yokoyama, T, Suzuki, R, Mizuguchi, M.
登録日2020-06-18
公開日2021-01-20
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Crystal structure of death-associated protein kinase 1 in complex with the dietary compound resveratrol.
Iucrj, 8, 2020
4YPD
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BU of 4ypd by Molmil
Crystal Structure of DAPK1 catalytic domain in complex with the hinge binding fragment 4-methylpyridazine
分子名称: 4-methylpyridazine, CHLORIDE ION, Death-associated protein kinase 1, ...
著者Grum-Tokars, V.L, Minasov, G, Roy, S.M, Anderson, W.F, Watterson, D.M.
登録日2015-03-12
公開日2015-05-13
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Crystal Structure of DAPK1 catalytic domain in complex with hinge binding fragments
To Be Published
5AV4
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BU of 5av4 by Molmil
Crystal structure of DAPK1-genistein complex in the presence of bromide ions.
分子名称: BROMIDE ION, Death-associated protein kinase 1, GENISTEIN
著者Yokoyama, T, Mizuguchi, M.
登録日2015-06-10
公開日2015-10-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.
J.Med.Chem., 58, 2015
3GU6
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BU of 3gu6 by Molmil
Crystal structure of DAPKQ23V-ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, Death-associated protein kinase 1
著者McNamara, L.K, Schavocky, J.S, Watterson, D.M, Brunzelle, J.S.
登録日2009-03-28
公開日2010-03-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Enzymatic activity and crystallographic analyses of a glycine-rich loop mutant of DAPK
To be Published
5AUV
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BU of 5auv by Molmil
Crystal structure of DAPK1 in complex with apigenin.
分子名称: 5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one, CHLORIDE ION, Death-associated protein kinase 1
著者Yokoyama, T, Mizuguchi, M.
登録日2015-06-10
公開日2015-10-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.
J.Med.Chem., 58, 2015
1JKS
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BU of 1jks by Molmil
1.5A X-RAY STRUCTURE OF APO FORM OF A CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE
分子名称: DEATH-ASSOCIATED PROTEIN KINASE
著者Tereshko, V, Teplova, M, Brunzelle, J, Watterson, D.M, Egli, M.
登録日2001-07-13
公開日2002-04-01
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal structures of the catalytic domain of human protein kinase associated with apoptosis and tumor suppression.
Nat.Struct.Biol., 8, 2001
5AV1
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BU of 5av1 by Molmil
Crystal structure of DAPK1 in the presence of bromide ions.
分子名称: BROMIDE ION, Death-associated protein kinase 1
著者Yokoyama, T, Mizuguchi, M.
登録日2015-06-10
公開日2015-10-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.
J.Med.Chem., 58, 2015
5AUW
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BU of 5auw by Molmil
Crystal structure of DAPK1 in complex with quercetin.
分子名称: 3,5,7,3',4'-PENTAHYDROXYFLAVONE, Death-associated protein kinase 1
著者Yokoyama, T, Mizuguchi, M.
登録日2015-06-10
公開日2015-10-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.
J.Med.Chem., 58, 2015
5AUX
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BU of 5aux by Molmil
Crystal structure of DAPK1 in complex with kaempferol.
分子名称: 3,5,7-TRIHYDROXY-2-(4-HYDROXYPHENYL)-4H-CHROMEN-4-ONE, CHLORIDE ION, Death-associated protein kinase 1
著者Yokoyama, T, Mizuguchi, M.
登録日2015-06-10
公開日2015-10-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.
J.Med.Chem., 58, 2015
5AV2
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BU of 5av2 by Molmil
Crystal structure of DAPK1-kaempferol complex in the presence of bromide ions.
分子名称: 3,5,7-TRIHYDROXY-2-(4-HYDROXYPHENYL)-4H-CHROMEN-4-ONE, BROMIDE ION, Death-associated protein kinase 1
著者Yokoyama, T, Mizuguchi, M.
登録日2015-06-10
公開日2015-10-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.502 Å)
主引用文献Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.
J.Med.Chem., 58, 2015
3EHA
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BU of 3eha by Molmil
Crystal structure of death associated protein kinase complexed with AMPPNP
分子名称: Death-associated protein kinase 1, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者McNamara, L.K, Watterson, D.M, Brunzelle, J.S.
登録日2008-09-11
公開日2009-04-28
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural insight into nucleotide recognition by human death-associated protein kinase.
Acta Crystallogr.,Sect.D, 65, 2009
4YO4
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BU of 4yo4 by Molmil
Crystal Structure of DAPK1 catalytic domain in complex with the hinge binding fragment phthalazine
分子名称: ACETATE ION, CHLORIDE ION, Death-associated protein kinase 1, ...
著者Grum-Tokars, V.L, Roy, S.M, Minasov, G, Anderson, W.F, Watterson, D.M.
登録日2015-03-11
公開日2015-05-06
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal Structure of DAPK1 catalytic domain in complex with hinge binding fragments
To Be Published
5AUZ
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BU of 5auz by Molmil
Crystal structure of DAPK1 in complex with genistein.
分子名称: Death-associated protein kinase 1, GENISTEIN
著者Yokoyama, T, Mizuguchi, M.
登録日2015-06-10
公開日2015-10-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.
J.Med.Chem., 58, 2015
3GU8
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BU of 3gu8 by Molmil
Crystal structure of DAPKL93G with N6-cyclopentyladenosine
分子名称: Death-associated protein kinase 1, N6-cyclopentyladenosine
著者McNamara, L.K, Schumacher, A.M, Schavocky, J.S, Watterson, D.M, Brunzelle, J.S.
登録日2009-03-28
公開日2010-03-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal structures of the DAPK gatekeeper mutant with N6-modified adenosine analogs.
To be Published
1JKL
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BU of 1jkl by Molmil
1.6A X-RAY STRUCTURE OF BINARY COMPLEX OF A CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE WITH ATP ANALOGUE
分子名称: DEATH-ASSOCIATED PROTEIN KINASE, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者Tereshko, V, Teplova, M, Brunzelle, J, Watterson, D.M, Egli, M.
登録日2001-07-12
公開日2002-04-01
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.62 Å)
主引用文献Crystal structures of the catalytic domain of human protein kinase associated with apoptosis and tumor suppression.
Nat.Struct.Biol., 8, 2001
7CCU
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BU of 7ccu by Molmil
Crystal structure of death-associated protein kinase 1 in complex with resveratrol
分子名称: Death-associated protein kinase 1, RESVERATROL, SULFATE ION
著者Yokoyama, T, Suzuki, R, Mizuguchi, M.
登録日2020-06-18
公開日2021-01-20
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.649 Å)
主引用文献Crystal structure of death-associated protein kinase 1 in complex with the dietary compound resveratrol.
Iucrj, 8, 2020
3GU5
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BU of 3gu5 by Molmil
Crystal structure of DAPKQ23V-AMPPNP-Mg2+
分子名称: Death-associated protein kinase 1, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者McNamara, L.K, Schavocky, J.S, Watterson, D.M, Brunzelle, J.S.
登録日2009-03-28
公開日2010-03-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Enzyme activity and crystallographic analyses of a glycine-rich loop mutant of DAPK
To be Published
3EH9
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BU of 3eh9 by Molmil
Crystal structure of death associated protein kinase complexed with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, Death-associated protein kinase 1, SULFATE ION
著者McNamara, L.K, Watterson, D.M, Brunzelle, J.S.
登録日2008-09-11
公開日2009-04-28
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural insight into nucleotide recognition by human death-associated protein kinase.
Acta Crystallogr.,Sect.D, 65, 2009
3DGK
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BU of 3dgk by Molmil
Crystal structure of a glycine-rich loop mutant of the death associated protein kinase catalytic domain
分子名称: Death-associated protein kinase 1
著者McNamara, L.K, Schavocky, J.P, Watterson, D.M, Brunzelle, J.S.
登録日2008-06-13
公開日2009-05-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献High resolution crystal structures of the death associated protein kinase catalytic domain with a key point mutation in the glycine-rich loop
To be Published
1YR5
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BU of 1yr5 by Molmil
1.7-A structure of calmodulin bound to a peptide from DAP kinase
分子名称: 19-mer from Death-associated protein kinase 1, CALCIUM ION, calmodulin
著者Kursula, P, Vahokoski, J, Wilmanns, M.
登録日2005-02-03
公開日2006-07-04
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Recognition of human death-associated protein kinases by calmodulin
To be Published
5AUU
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BU of 5auu by Molmil
Crystal structure of DAPK1 in complex with luteolin.
分子名称: 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4-one, Death-associated protein kinase 1
著者Yokoyama, T, Mizuguchi, M.
登録日2015-06-10
公開日2015-10-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.
J.Med.Chem., 58, 2015

 

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