5UWW
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6M60
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![BU of 6m60 by Molmil](/molmil-images/mine/6m60) | Plumbagin in complex with CRM1#-Ran-RanBP1 | 分子名称: | (2~{R})-2-methyl-5-oxidanyl-2,3-dihydronaphthalene-1,4-dione, CHLORIDE ION, DIMETHYL SULFOXIDE, ... | 著者 | Sun, Q, Lei, Y. | 登録日 | 2020-03-12 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | Novel Mechanistic Observations and NES-Binding Groove Features Revealed by the CRM1 Inhibitors Plumbagin and Oridonin. J.Nat.Prod., 84, 2021
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6XJU
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![BU of 6xju by Molmil](/molmil-images/mine/6xju) | Crystal Structure of KPT-8602 bound to CRM1 (E582K, 537-DLTVK-541 to GLCEQ) | 分子名称: | (2R)-3-{3-[3,5-bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}-2-(pyrimidin-5-yl)propanamide, Exportin-1, GTP-binding nuclear protein Ran, ... | 著者 | Baumhardt, J.M, Chook, Y.M. | 登録日 | 2020-06-24 | 公開日 | 2021-01-27 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.193 Å) | 主引用文献 | Recurrent XPO1 mutations alter pathogenesis of chronic lymphocytic leukemia. J Hematol Oncol, 14, 2021
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6X2U
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4HB0
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![BU of 4hb0 by Molmil](/molmil-images/mine/4hb0) | Crystal structure of CRM1 inhibitor Leptomycin B in complex with CRM1(K541Q,K542Q,R543S,K545Q,K548Q,K579Q)-Ran-RanBP1 | 分子名称: | CHLORIDE ION, Exportin-1, GTP-binding nuclear protein Ran, ... | 著者 | Sun, Q, Chook, Y.M. | 登録日 | 2012-09-27 | 公開日 | 2013-01-09 | 最終更新日 | 2017-07-26 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Nuclear export inhibition through covalent conjugation and hydrolysis of Leptomycin B by CRM1. Proc.Natl.Acad.Sci.USA, 110, 2013
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4GPT
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![BU of 4gpt by Molmil](/molmil-images/mine/4gpt) | Crystal structure of KPT251 in complex with CRM1-Ran-RanBP1 | 分子名称: | 1,2-ETHANEDIOL, 2-(2-{3-[3,5-bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}ethyl)-1,3,4-oxadiazole, CHLORIDE ION, ... | 著者 | Sun, Q, Chook, Y.M. | 登録日 | 2012-08-21 | 公開日 | 2012-09-05 | 最終更新日 | 2013-01-23 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | Antileukemic activity of nuclear export inhibitors that spare normal hematopoietic cells. Leukemia, 27, 2013
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5UWJ
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5UWR
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![BU of 5uwr by Molmil](/molmil-images/mine/5uwr) | |
5UWU
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![BU of 5uwu by Molmil](/molmil-images/mine/5uwu) | |
8HQ5
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![BU of 8hq5 by Molmil](/molmil-images/mine/8hq5) | G6 in complex with CRM1-Ran-RanBP1 | 分子名称: | 3-[(4-bromophenyl)carbonylamino]-4-[4-(5-chloranyl-2-methyl-phenyl)piperazin-1-yl]benzoic acid, 3[N-MORPHOLINO]PROPANE SULFONIC ACID, CHLORIDE ION, ... | 著者 | Sun, Q, Lei, Y. | 登録日 | 2022-12-13 | 公開日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | F1 in complex with CRM1-Ran-RanBP1 To Be Published
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5UWH
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5UWQ
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![BU of 5uwq by Molmil](/molmil-images/mine/5uwq) | |
5DI9
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4HAX
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![BU of 4hax by Molmil](/molmil-images/mine/4hax) | |
5DHF
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![BU of 5dhf by Molmil](/molmil-images/mine/5dhf) | |
8HUF
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![BU of 8huf by Molmil](/molmil-images/mine/8huf) | B28 in complex with CRM1-Ran-RanBP1 | 分子名称: | 3-[(4-chlorophenyl)carbonylamino]-4-[4-(2,5-dimethylphenyl)piperazin-1-yl]benzoic acid, BROMIDE ION, CHLORIDE ION, ... | 著者 | Sun, Q, Lei, Y. | 登録日 | 2022-12-23 | 公開日 | 2023-12-27 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (2.29 Å) | 主引用文献 | Discovery of a Hidden Pocket beneath the NES Groove by Novel Noncovalent CRM1 Inhibitors. J.Med.Chem., 66, 2023
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6X2R
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![BU of 6x2r by Molmil](/molmil-images/mine/6x2r) | |
5YSU
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![BU of 5ysu by Molmil](/molmil-images/mine/5ysu) | |
5YTB
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8ITV
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![BU of 8itv by Molmil](/molmil-images/mine/8itv) | KL2.1 in complex with CRM1-Ran-RanBP1 | 分子名称: | (3~{S},5~{R},6~{E},8~{Z},10~{R},12~{E},14~{E},16~{S})-3,16-bis(azanyl)-8,10,12-trimethyl-16-[(2~{S},4~{R},5~{S},6~{S})-5-methyl-4-oxidanyl-6-[(~{E})-prop-1-enyl]oxan-2-yl]-5-oxidanyl-hexadeca-6,8,12,14-tetraenoic acid, ACETATE ION, CHLORIDE ION, ... | 著者 | Sun, Q, Jian, L. | 登録日 | 2023-03-23 | 公開日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | KL2.1 in complex with CRM1-Ran-RanBP1 To Be Published
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6A3A
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![BU of 6a3a by Molmil](/molmil-images/mine/6a3a) | MVM NES mutant Nm2 in complex with CRM1-Ran-RanBP1 | 分子名称: | 1,2-ETHANEDIOL, Exportin-1, GLYCEROL, ... | 著者 | Sun, Q, Li, Y. | 登録日 | 2018-06-15 | 公開日 | 2019-06-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor. Int J Nanomedicine, 16, 2021
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4HAY
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![BU of 4hay by Molmil](/molmil-images/mine/4hay) | Crystal structure of CRM1 inhibitor Leptomycin B in complex with CRM1(K548E,K579Q)-Ran-RanBP1 | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, Exportin-1, ... | 著者 | Sun, Q, Chook, Y.M. | 登録日 | 2012-09-27 | 公開日 | 2013-01-09 | 最終更新日 | 2017-07-26 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Nuclear export inhibition through covalent conjugation and hydrolysis of Leptomycin B by CRM1. Proc.Natl.Acad.Sci.USA, 110, 2013
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6X2Y
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5UWT
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![BU of 5uwt by Molmil](/molmil-images/mine/5uwt) | |
5UWO
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![BU of 5uwo by Molmil](/molmil-images/mine/5uwo) | |