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PDB: 10 件

1FAS
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1.9 ANGSTROM RESOLUTION STRUCTURE OF FASCICULIN 1, AN ANTI-ACETYLCHOLINESTERASE TOXIN FROM GREEN MAMBA SNAKE VENOM
分子名称: FASCICULIN 1
著者Le Du, M.H, Marchot, P, Bougis, P.E, Fontecilla-Camps, J.C.
登録日1992-08-07
公開日1993-10-31
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献1.9-A resolution structure of fasciculin 1, an anti-acetylcholinesterase toxin from green mamba snake venom.
J.Biol.Chem., 267, 1992
1FSC
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Crystal Structure of Fasciculin 2 from Green Mamba Snake Venom: Evidence for Unusual Loop Flexibility
分子名称: FASCICULIN 2, UNKNOWN LIGAND
著者Housset, D, Le Du, M.H, Fontecilla-Camps, J.C.
登録日1995-03-27
公開日1995-07-10
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of fasciculin 2 from green mamba snake venom: evidence for unusual loop flexibility.
Acta Crystallogr.,Sect.D, 52, 1996
1KU6
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Fasciculin 2-Mouse Acetylcholinesterase Complex
分子名称: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, ...
著者Bourne, Y, Burmeister, W, Taylor, P, Marchot, P.
登録日2002-01-21
公開日2003-12-23
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural insights into ligand interactions at the acetylcholinesterase peripheral anionic site.
EMBO J., 22, 2003
4EY8
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Crystal structure of recombinant human acetylcholinesterase in complex with fasciculin-2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Acetylcholinesterase, Fasciculin-2, ...
著者Cheung, J, Rudolph, M, Burshteyn, F, Cassidy, M, Gary, E, Love, J, Height, J, Franklin, M.
登録日2012-05-01
公開日2012-10-17
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.5958 Å)
主引用文献Structures of human acetylcholinesterase in complex with pharmacologically important ligands.
J.Med.Chem., 55, 2012
1B41
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HUMAN ACETYLCHOLINESTERASE COMPLEXED WITH FASCICULIN-II, GLYCOSYLATED PROTEIN
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, ...
著者Kryger, G, Harel, M, Shafferman, A, Silman, I, Sussman, J.L.
登録日1999-01-05
公開日2001-01-17
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.76 Å)
主引用文献Structures of recombinant native and E202Q mutant human acetylcholinesterase complexed with the snake-venom toxin fasciculin-II.
Acta Crystallogr.,Sect.D, 56, 2000
1F8U
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CRYSTAL STRUCTURE OF MUTANT E202Q OF HUMAN ACETYLCHOLINESTERASE COMPLEXED WITH GREEN MAMBA VENOM PEPTIDE FASCICULIN-II
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, FASCICULIN II
著者Kryger, G, Harel, M, Shafferman, A, Silman, I, Sussman, J.L.
登録日2000-07-05
公開日2001-01-17
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structures of recombinant native and E202Q mutant human acetylcholinesterase complexed with the snake-venom toxin fasciculin-II.
Acta Crystallogr.,Sect.D, 56, 2000
2X8B
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Crystal structure of human acetylcholinesterase inhibited by aged tabun and complexed with fasciculin-II
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETHYLCHOLINESTERASE, CHLORIDE ION, ...
著者Carletti, E, Colletier, J.P, Nachon, F.
登録日2010-03-08
公開日2010-04-28
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Structural evidence that human acetylcholinesterase inhibited by tabun ages through O-dealkylation.
J. Med. Chem., 53, 2010
1FSS
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ACETYLCHOLINESTERASE (E.C. 3.1.1.7) COMPLEXED WITH FASCICULIN-II
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, FASCICULIN II, ...
著者Harel, M, Kleywegt, G.J, Silman, I, Sussman, J.L.
登録日1995-10-25
公開日1996-03-08
最終更新日2021-06-02
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal structure of an acetylcholinesterase-fasciculin complex: interaction of a three-fingered toxin from snake venom with its target.
Structure, 3, 1995
4BDT
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Human acetylcholinesterase in complex with huprine W and fasciculin 2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, CHLORIDE ION, ...
著者Nachon, F, Carletti, E, Ronco, C, Trovaslet, M, Nicolet, Y, Jean, L, Renard, P.-Y.
登録日2012-10-06
公開日2013-05-29
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.104 Å)
主引用文献Crystal structures of human cholinesterases in complex with huprine W and tacrine: elements of specificity for anti-Alzheimer's drugs targeting acetyl- and butyryl-cholinesterase.
Biochem. J., 453, 2013
1MAH
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FASCICULIN2-MOUSE ACETYLCHOLINESTERASE COMPLEX
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, FASCICULIN 2
著者Bourne, Y, Taylor, P, Marchot, P.
登録日1995-11-21
公開日1996-04-03
最終更新日2021-03-31
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Acetylcholinesterase inhibition by fasciculin: crystal structure of the complex.
Cell(Cambridge,Mass.), 83, 1995

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