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PDB: 55 件

1R6J
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Ultrahigh resolution Crystal Structure of syntenin PDZ2
分子名称: CHLORIDE ION, Syntenin 1
著者Kang, B.S, Devedjiev, Y, Derewenda, U, Derewenda, Z.S.
登録日2003-10-15
公開日2004-05-04
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (0.73 Å)
主引用文献The PDZ2 domain of syntenin at ultra-high resolution: bridging the gap between small molecule and macromolecular crystal chemistry
J.Mol.Biol., 338, 2004
1NTE
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BU of 1nte by Molmil
CRYSTAL STRUCTURE ANALYSIS OF THE SECOND PDZ DOMAIN OF SYNTENIN
分子名称: OXYGEN ATOM, Syntenin 1
著者Kang, B.S, Cooper, D.R, Devedjiev, Y, Derewenda, U, Derewenda, Z.S.
登録日2003-01-29
公開日2003-07-15
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.24 Å)
主引用文献Molecular roots of degenerate specificity in syntenin's PDZ2 domain: reassessment of the PDZ recognition paradigm.
Structure, 11, 2003
1OBX
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Crystal structure of the complex of PDZ2 of syntenin with an interleukin 5 receptor alpha peptide.
分子名称: COBALT (II) ION, INTERLEUKIN 5 RECEPTOR ALPHA, SULFATE ION, ...
著者Kang, B.S, Cooper, D.R, Devedjiev, Y, Derewenda, U, Derewenda, Z.S.
登録日2003-01-31
公開日2003-07-10
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Molecular Roots of Degenerate Specificity in Syntenin'S Pdz2 Domain: Reassessment of the Pdz Recognition Paradigm
Structure, 11, 2003
8BLU
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BU of 8blu by Molmil
The PDZ domains of human SDCBP
分子名称: 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Daniel-Mozo, M, Bountra, C, von Delft, F, Brennan, P.E.
登録日2022-11-10
公開日2022-11-30
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The PDZ domains of human SDCBP
To Be Published
8BLV
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BU of 8blv by Molmil
The PDZ domains of human SDCBP with a bound SDC4 C-terminal peptide
分子名称: 1,2-ETHANEDIOL, SULFATE ION, Syndecan-4, ...
著者Bradshaw, W.J, Katis, V.L, Daniel-Mozo, M, Bountra, C, von Delft, F, Brennan, P.E.
登録日2022-11-10
公開日2022-12-21
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The PDZ domains of human SDCBP with a bound SDC4 C-terminal peptide
To Be Published
1W9E
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BU of 1w9e by Molmil
Crystal structure of the PDZ tandem of human syntenin in complex with TNEFYF peptide
分子名称: BENZOIC ACID, SYNTENIN 1, TNEFYF PEPTIDE
著者Grembecka, J, Cierpicki, T, Devedjiev, Y, Cooper, D.R, Derewenda, U, Derewenda, Z.S.
登録日2004-10-09
公開日2006-03-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献The Binding of the Pdz Tandem of Syntenin to Target Proteins.
Biochemistry, 45, 2006
1OBZ
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BU of 1obz by Molmil
Crystal structure of the complex of the PDZ tandem of syntenin with an interleukin 5 receptor alpha peptide.
分子名称: ACETATE ION, INTERLEUKIN 5 RECEPTOR ALPHA, SYNTENIN 1
著者Kang, B.S, Cooper, D.R, Devedjiev, Y, Derewenda, U, Derewenda, Z.S.
登録日2003-01-31
公開日2003-07-11
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Molecular Roots of Degenerate Specificity in Syntenin'S Pdz2 Domain: Reassessment of the Pdz Recognition Paradigm
Structure, 11, 2003
1W9Q
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BU of 1w9q by Molmil
Crystal structure of the PDZ tandem of human syntenin in complex with TNEFAF peptide
分子名称: BENZOIC ACID, SYNTENIN 1, TNEFAF PEPTIDE
著者Grembecka, J, Cierpicki, T, Devedjiev, Y, Cooper, D.R, Derewenda, Z.S.
登録日2004-10-15
公開日2006-03-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The Binding of the Pdz Tandem of Syntenin to Target Proteins.
Biochemistry, 45, 2006
7FT9
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BU of 7ft9 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z45636695
分子名称: 1,2-ETHANEDIOL, 4-[(METHYLSULFONYL)AMINO]BENZOIC ACID, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT5
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BU of 7ft5 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with POB0093
分子名称: 1,2-ETHANEDIOL, 4-(4-methoxyphenyl)oxane-4-carboxylic acid, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT7
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BU of 7ft7 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z57127349
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
1V1T
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BU of 1v1t by Molmil
Crystal structure of the PDZ tandem of human syntenin in complex with TNEYKV peptide
分子名称: BENZOIC ACID, SYNTENIN 1, TNEYKV PEPTIDE
著者Grembecka, J, Cierpicki, T, Devedjiev, Y, Cooper, D.R, Derewenda, U, Derewenda, Z.S.
登録日2004-04-23
公開日2005-06-14
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The Binding of the Pdz Tandem of Syntenin to Target Proteins.
Biochemistry, 45, 2006
7FTD
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BU of 7ftd by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z27782662
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
1OBY
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BU of 1oby by Molmil
Crystal structure of the complex of PDZ2 of syntenin with a syndecan-4 peptide.
分子名称: SULFATE ION, SYNDECAN-4, SYNTENIN 1
著者Kang, B.S, Cooper, D.R, Devedjiev, Y, Derewenda, U, Derewenda, Z.S.
登録日2003-01-31
公開日2003-07-11
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Molecular Roots of Degenerate Specificity in Syntenin'S Pdz2 Domain: Reassessment of the Pdz Recognition Paradigm
Structure, 11, 2003
7FT6
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BU of 7ft6 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with POB0008
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSP
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BU of 7fsp by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1650168321
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FTC
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BU of 7ftc by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1509711879
分子名称: 1,2-ETHANEDIOL, 6-bromo-7-hydroxy-2,2-dimethyl-2H,4H-1,3-benzodioxin-4-one, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSO
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BU of 7fso by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z198195770
分子名称: 1,2-ETHANEDIOL, D-GLUTAMIC ACID, GLYCINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSX
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BU of 7fsx by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1328078283
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
1N99
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BU of 1n99 by Molmil
CRYSTAL STRUCTURE OF THE PDZ TANDEM OF HUMAN SYNTENIN
分子名称: Syntenin 1
著者Kang, B.S, Cooper, D.R, Jelen, F, Devedjiev, Y, Derewenda, U, Dauter, Z, Otlewski, J, Derewenda, Z.S.
登録日2002-11-22
公開日2003-04-15
最終更新日2022-12-21
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献PDZ Tandem of Human Syntenin: Crystal Structure and Functional Properties
Structure, 11, 2003
7FSJ
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BU of 7fsj by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z57744712
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSU
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BU of 7fsu by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z729726784
分子名称: 1,2-ETHANEDIOL, 2-cyclopentyl-N-(3-methyl-1,2,4-oxadiazol-5-yl)acetamide, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FST
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BU of 7fst by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z26968795
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
6R9H
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BU of 6r9h by Molmil
Crystal structure of the PDZ tandem of syntenin in complex with fragment C58
分子名称: (2~{S})-2-[2-(4-chlorophenyl)sulfanylethanoylamino]-3-methyl-butanoic acid, ACETATE ION, PHOSPHATE ION, ...
著者Feracci, M, Barral, K.
登録日2019-04-03
公開日2021-02-03
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Pharmacological inhibition of syntenin PDZ2 domain impairs breast cancer cell activities and exosome loadifing with syndecan and EpCAM cargo.
J Extracell Vesicles, 10, 2020
8HCK
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BU of 8hck by Molmil
NMR fragment-based screening against the two PDZ do-mains of MDA-9
分子名称: 4-BUTYL-1,2-DIPHENYL-PYRAZOLIDINE-3,5-DIONE, GLYCEROL, SULFATE ION, ...
著者Tang, H.
登録日2022-11-01
公開日2023-11-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献NMR fragment-based screening against the two PDZ do-mains of MDA-9
To Be Published

 

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