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PDB: 1 件

9B4U
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BU of 9b4u by Molmil
Crystal structure of p110alpha-RBD covalently bound to a breaker compound BBO-10203 via Cys242
分子名称: 1-[(4R,8R)-2-[(4M,7P)-7-[2,4-difluoro-6-(2-methoxyethoxy)phenyl]-4-(1-methyl-1H-indazol-5-yl)thieno[3,2-c]pyridin-6-yl]-4-methyl-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]propan-1-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
著者Czyzyk, D.J, Simanshu, D.K.
登録日2024-03-21
公開日2025-06-25
実験手法X-RAY DIFFRACTION (2.21 Å)
主引用文献BBO-10203 inhibits tumor growth without inducing hyperglycemia by blocking RAS-PI3K alpha interaction.
Science, 2025

238582

件を2025-07-09に公開中

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