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PDB: 4 件

6CYG
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BU of 6cyg by Molmil
Hsp90-alpha N-domain bound to NEOCA
分子名称: 5'-N-(2-HYDROXYL)ETHYL CARBOXYAMIDO ADENOSINE, Heat shock protein HSP 90-alpha, MAGNESIUM ION
著者Huck, J.D, Campomizzi, C, Gewirth, D.T.
登録日2018-04-05
公開日2019-04-10
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.503922 Å)
主引用文献NECA derivatives exploit the paralog-specific properties of the site 3 side pocket of Grp94, the endoplasmic reticulum Hsp90.
J.Biol.Chem., 294, 2019
6D1X
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BU of 6d1x by Molmil
N-Domain Of Grp94, with the Charged Domain, In Complex With the Novel Ligand N-Propyl Carboxyamido Adenosine
分子名称: Endoplasmin, N-PROPYL CARBOXYAMIDO ADENOSINE, TETRAETHYLENE GLYCOL
著者Gewirth, D.T, Immormino, R.M.
登録日2018-04-12
公開日2018-05-02
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献NECA derivatives exploit the paralog-specific properties of the site 3 side pocket of Grp94, the endoplasmic reticulum Hsp90.
J.Biol.Chem., 294, 2019
6CYH
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BU of 6cyh by Molmil
Hsp90-alpha N-domain bound to NEACA
分子名称: 5'-N-[(2-AMINO)ETHYL CARBOXAMIDO] ADENOSINE, Heat shock protein HSP 90-alpha, MAGNESIUM ION
著者Huck, J.D, Campomizzi, C, Gewirth, D.T.
登録日2018-04-05
公開日2019-04-10
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献NECA derivatives exploit the paralog-specific properties of the site 3 side pocket of Grp94, the endoplasmic reticulum Hsp90.
J.Biol.Chem., 294, 2019
6CYI
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BU of 6cyi by Molmil
Grp94 N-domain bound to NEOCA
分子名称: 5'-N-(2-HYDROXYL)ETHYL CARBOXYAMIDO ADENOSINE, Endoplasmin, TETRAETHYLENE GLYCOL, ...
著者Huck, J.D, Aw, W.J, Gewirth, D.T.
登録日2018-04-05
公開日2019-04-10
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.7565825 Å)
主引用文献NECA derivatives exploit the paralog-specific properties of the site 3 side pocket of Grp94, the endoplasmic reticulum Hsp90.
J.Biol.Chem., 294, 2019

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件を2024-07-17に公開中

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