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PDB: 4 件

6SGK
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BU of 6sgk by Molmil
Nek2 kinase bound to inhibitor 102
分子名称: 2-phenylazanyl-9~{H}-purine-6-carbonitrile, Serine/threonine-protein kinase Nek2
著者Richards, M.W, Mas-Droux, C.P, Bayliss, R.
登録日2019-08-05
公開日2020-06-17
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献2-Arylamino-6-ethynylpurines are cysteine-targeting irreversible inhibitors of Nek2 kinase.
Rsc Med Chem, 11, 2020
6SGD
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BU of 6sgd by Molmil
Nek2 kinase covalently bound to 2-arylamino-6-ethynylpurine inhibitor 24
分子名称: 4-[(6-ethenyl-7~{H}-purin-2-yl)amino]benzenesulfonamide, CHLORIDE ION, SODIUM ION, ...
著者Richards, M.W, Mas-Droux, C.P, Bayliss, R.
登録日2019-08-04
公開日2020-06-17
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献2-Arylamino-6-ethynylpurines are cysteine-targeting irreversible inhibitors of Nek2 kinase.
Rsc Med Chem, 11, 2020
6SGI
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BU of 6sgi by Molmil
Nek2 kinase bound to inhibitor 96
分子名称: 4-[(6-ethyl-7~{H}-purin-2-yl)amino]benzenesulfonamide, CHLORIDE ION, Serine/threonine-protein kinase Nek2
著者Richards, M.W, Mas-Droux, C.P, Bayliss, R.
登録日2019-08-05
公開日2020-06-17
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献2-Arylamino-6-ethynylpurines are cysteine-targeting irreversible inhibitors of Nek2 kinase.
Rsc Med Chem, 11, 2020
6SGH
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BU of 6sgh by Molmil
Nek2 kinase covalently bound to 2-arylamino-6-ethynylpurine inhibitor 66
分子名称: 2-[4-[(6-ethenyl-9~{H}-purin-2-yl)amino]phenyl]ethanamide, Serine/threonine-protein kinase Nek2
著者Richards, M.W, Mas-Droux, C.P, Bayliss, R.
登録日2019-08-04
公開日2020-06-17
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献2-Arylamino-6-ethynylpurines are cysteine-targeting irreversible inhibitors of Nek2 kinase.
Rsc Med Chem, 11, 2020

222624

件を2024-07-17に公開中

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