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PDB: 4 件

7Z9M
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BU of 7z9m by Molmil
E.coli gyrase holocomplex with 217 bp DNA and Albi-1 (site AA)
分子名称: 4-[[4-[[5-[[(2S)-2-[[5-[(4-cyanophenyl)carbonylamino]pyridin-2-yl]carbonylamino]-3-(1H-1,2,3-triazol-4-yl)propanoyl]amino]pyridin-2-yl]carbonylamino]-2-oxidanyl-3-propan-2-yloxy-phenyl]carbonylamino]benzoic acid, DNA (5'-D(*AP*AP*TP*CP*AP*CP*CP*CP*GP*CP*AP*CP*AP*GP*AP*TP*TP*T)-3'), DNA (5'-D(*GP*AP*TP*TP*TP*TP*AP*TP*GP*CP*CP*TP*GP*AP*TP*TP*CP*T)-3'), ...
著者Ghilarov, D, Heddle, J.G.H.
登録日2022-03-21
公開日2023-02-15
最終更新日2023-07-19
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin.
Nat Catal, 6, 2023
7Z9G
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BU of 7z9g by Molmil
E.coli gyrase holocomplex with 217 bp DNA and Albi-2
分子名称: 4-[[3-(2-azanylethoxy)-2-oxidanyl-4-[[5-[[(2~{S})-2-[[4-[(6-oxidanylnaphthalen-2-yl)carbonylamino]phenyl]carbonylamino]-3-(1~{H}-1,2,3-triazol-4-yl)propanoyl]amino]pyridin-2-yl]carbonylamino]phenyl]carbonylamino]-3-methoxy-2-oxidanyl-benzoic acid, DNA (5'-D(*AP*AP*TP*CP*AP*CP*CP*CP*GP*CP*AP*CP*AP*GP*AP*TP*TP*T)-3'), DNA (5'-D(*GP*AP*TP*TP*TP*TP*AP*TP*GP*CP*CP*TP*GP*AP*TP*TP*CP*T)-3'), ...
著者Ghilarov, D, Heddle, J.G.H.
登録日2022-03-21
公開日2023-02-15
最終更新日2023-07-19
実験手法ELECTRON MICROSCOPY (3.25 Å)
主引用文献Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin.
Nat Catal, 6, 2023
7Z9C
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BU of 7z9c by Molmil
E.coli gyrase holocomplex with 217 bp DNA and albicidin
分子名称: DNA (5'-D(*AP*AP*TP*CP*AP*CP*CP*CP*GP*CP*AP*CP*AP*GP*AP*TP*TP*T)-3'), DNA (5'-D(*GP*AP*TP*TP*TP*TP*AP*TP*GP*CP*CP*TP*GP*AP*TP*TP*CP*T)-3'), DNA (5'-D(P*AP*AP*AP*TP*CP*TP*GP*TP*GP*CP*GP*GP*GP*T)-3'), ...
著者Ghilarov, D, Heddle, J.G.H, Suessmuth, R.
登録日2022-03-21
公開日2023-02-15
最終更新日2023-07-19
実験手法ELECTRON MICROSCOPY (3.06 Å)
主引用文献Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin.
Nat Catal, 6, 2023
7Z9K
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BU of 7z9k by Molmil
E.coli gyrase holocomplex with 217 bp DNA and Albi-1 (site TG)
分子名称: 4-[[4-[[5-[[(2S)-2-[[5-[(4-cyanophenyl)carbonylamino]pyridin-2-yl]carbonylamino]-3-(1H-1,2,3-triazol-4-yl)propanoyl]amino]pyridin-2-yl]carbonylamino]-2-oxidanyl-3-propan-2-yloxy-phenyl]carbonylamino]benzoic acid, DNA (5'-D(*AP*AP*TP*CP*AP*CP*CP*CP*GP*CP*AP*CP*AP*GP*AP*TP*TP*T)-3'), DNA (5'-D(*GP*AP*TP*TP*TP*TP*AP*TP*GP*CP*CP*TP*GP*AP*TP*TP*CP*T)-3'), ...
著者Ghilarov, D, Heddle, J.G.H.
登録日2022-03-21
公開日2023-03-08
最終更新日2023-07-19
実験手法ELECTRON MICROSCOPY (3.25 Å)
主引用文献Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin.
Nat Catal, 6, 2023

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件を2024-06-12に公開中

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