PDB クエリの検索結果 - 日本蛋白質構造データバンク

PDB: 3 件

BRD4 Bromodomain 1 in complex with multi-action inhibitor SRX3212P
分子名称:	7-[7-oxo-5-(piperazin-1-yl)-7H-thieno[3,2-b]pyran-3-yl]-N-[(pyridin-3-yl)methyl]-2,3-dihydro-1,4-benzodioxine-5-carboxamide, Bromodomain-containing protein 4
著者	Vann, K.R, Kutateladze, T.G.
登録日	2020-05-29
公開日	2020-08-05
最終更新日	2023-10-18
実験手法	X-RAY DIFFRACTION (1.951 Å)
主引用文献	Design of thienopyranone-based BET inhibitors that bind multiple synthetic lethality targets. Sci Rep, 10, 2020

BRD4 Bromodomain 1 in complex with multi-action inhibitor SRX3212
分子名称:	7-[5-(morpholin-4-yl)-7-oxo-7H-thieno[3,2-b]pyran-3-yl]-N-[(pyridin-3-yl)methyl]-2,3-dihydro-1,4-benzodioxine-5-carboxamide, Bromodomain-containing protein 4
著者	Vann, K.R, Kutateladze, T.G.
登録日	2020-05-29
公開日	2020-08-05
最終更新日	2023-10-18
実験手法	X-RAY DIFFRACTION (2.7 Å)
主引用文献	Design of thienopyranone-based BET inhibitors that bind multiple synthetic lethality targets. Sci Rep, 10, 2020

BRD4 Bromodomain 1 in complex with multi-action inhibitor SF2523P
分子名称:	3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(piperazin-1-yl)-7H-thieno[3,2-b]pyran-7-one, Bromodomain-containing protein 4
著者	Vann, K.R, Kutateladze, T.G.
登録日	2020-05-29
公開日	2020-08-05
最終更新日	2023-10-18
実験手法	X-RAY DIFFRACTION (2.5 Å)
主引用文献	Design of thienopyranone-based BET inhibitors that bind multiple synthetic lethality targets. Sci Rep, 10, 2020