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PDB: 1 件

6TD3
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Structure of DDB1 bound to CR8-engaged CDK12-cyclinK
分子名称: (2R)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9H-purin-2-yl}amino)butan-1-ol, Cyclin-K, Cyclin-dependent kinase 12, ...
著者Bunker, R.D, Petzold, G, Kozicka, Z, Thoma, N.H.
登録日2019-11-07
公開日2020-06-17
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.46 Å)
主引用文献The CDK inhibitor CR8 acts as a molecular glue degrader that depletes cyclin K.
Nature, 585, 2020

222926

件を2024-07-24に公開中

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