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PDB: 1 件

4WIV
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BU of 4wiv by Molmil
Crystal Structure of the first bromodomain of human BRD4 in complex with a novel inhibitor UMB32 (N-TERT-BUTYL-2-[4-(3,5-DIMETHYL-1,2-OXAZOL-4-YL) PHENYL]IMIDAZO[1,2-A]PYRAZIN-3-AMINE)
分子名称: 1,2-ETHANEDIOL, Bromodomain-containing protein 4, GLYCEROL, ...
著者Xu, X, Blacklow, S.
登録日2014-09-26
公開日2014-10-29
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Biased multicomponent reactions to develop novel bromodomain inhibitors.
J.Med.Chem., 57, 2014

222926

件を2024-07-24に公開中

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