4MUW
| Crystal Structure of PDE10A with Novel Keto-Benzimidazole Inhibitor | 分子名称: | 2-{4-[(6,7-difluoro-1H-benzimidazol-2-yl)amino]phenoxy}-N-methyl-3,4'-bipyridin-2'-amine, GLYCEROL, SULFATE ION, ... | 著者 | Chmait, S, Jordan, S. | 登録日 | 2013-09-23 | 公開日 | 2013-10-23 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.639 Å) | 主引用文献 | Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A). J.Med.Chem., 56, 2013
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4MVH
| Crystal Structure of PDE10A with Novel Keto-Benzimidazole Inhibitor | 分子名称: | 1H-benzimidazol-2-yl(4-{[3-(morpholin-4-yl)pyrazin-2-yl]oxy}phenyl)methanone, SULFATE ION, ZINC ION, ... | 著者 | Chmait, S, Jordan, S. | 登録日 | 2013-09-24 | 公開日 | 2013-10-23 | 最終更新日 | 2014-01-15 | 実験手法 | X-RAY DIFFRACTION (2.496 Å) | 主引用文献 | Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A). J.Med.Chem., 56, 2013
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