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PDB: 1 件

5T0L
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Crystal structure of Toxoplasma gondii TS-DHFR complexed with NADPH, dUMP, PDDF and 5-(4-(3,4-dichlorophenyl)piperazin-1-yl)pyrimidine-2,4-diamine (TRC-15)
分子名称: 10-PROPARGYL-5,8-DIDEAZAFOLIC ACID, 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, 5-[4-(3,4-dichlorophenyl)piperazin-1-yl]pyrimidine-2,4-diamine, ...
著者Thomas, S.B, Chen, Z, Lu, H, Li, Y.
登録日2016-08-16
公開日2016-09-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.13 Å)
主引用文献Discovery of Potent and Selective Leads against Toxoplasma gondii Dihydrofolate Reductase via Structure-Based Design.
ACS Med Chem Lett, 7, 2016

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件を2024-07-17に公開中

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