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PDB: 1 件

8XKP
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Crystal structure of human tyrosine-protein kinase Fes/Fps in complex with compound 17c
分子名称: 7-[[(1R,2S)-2-azanylcyclohexyl]amino]-5-[[3-[(2S,6R)-2,6-dimethylmorpholin-4-yl]phenyl]amino]-4-oxidanylidene-3H-pyrido[3,4-d]pyridazine-8-carbonitrile, SULFATE ION, Tyrosine-protein kinase Fes/Fps
著者Baba, D, Hanzawa, H.
登録日2023-12-23
公開日2025-01-01
最終更新日2025-03-19
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Optimization of Novel Pyrido-pyridazinone Derivatives as FER Tyrosine Kinase Inhibitors, Leading to the Potent DS08701581.
Acs Med.Chem.Lett., 15, 2024

238582

件を2025-07-09に公開中

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