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PDB: 2 件

6RFJ
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BU of 6rfj by Molmil
IRAK4 IN COMPLEX WITH inhibitor
分子名称: Interleukin-1 receptor-associated kinase 4, SULFATE ION, methyl 4-[4-[[6-(cyanomethyl)-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-4-yl]amino]cyclohexyl]piperazine-1-carboxylate
著者Xue, Y, Degorce, S.L, Robb, G.R, Ferguson, A.D.
登録日2019-04-15
公開日2019-10-30
最終更新日2019-11-27
実験手法X-RAY DIFFRACTION (2.61 Å)
主引用文献Discovery of a Series of 5-Azaquinazolines as Orally Efficacious IRAK4 Inhibitors Targeting MyD88L265PMutant Diffuse Large B Cell Lymphoma.
J.Med.Chem., 62, 2019
6RFI
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BU of 6rfi by Molmil
IRAK4 IN COMPLEX WITH inhibitor
分子名称: Interleukin-1 receptor-associated kinase 4, SULFATE ION, methyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylate
著者Xue, Y, Degorce, S.L, Robb, G.R, Ferguson, A.D.
登録日2019-04-15
公開日2019-10-30
最終更新日2019-11-27
実験手法X-RAY DIFFRACTION (2.31 Å)
主引用文献Discovery of a Series of 5-Azaquinazolines as Orally Efficacious IRAK4 Inhibitors Targeting MyD88L265PMutant Diffuse Large B Cell Lymphoma.
J.Med.Chem., 62, 2019

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件を2024-07-17に公開中

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