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PDB: 1 件

6B0F
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ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH LSZ102
分子名称: Estrogen receptor, GLYCEROL, LSZ102
著者Kirby, C.A, Baird, J.
登録日2017-09-14
公開日2018-04-04
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.86 Å)
主引用文献Discovery of LSZ102, a Potent, Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) for the Treatment of Estrogen Receptor Positive Breast Cancer.
J. Med. Chem., 61, 2018

222926

件を2024-07-24に公開中

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