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PDB: 1 件

4Z16
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Crystal Structure of the Jak3 Kinase Domain Covalently Bound to N-(3-(((5-chloro-2-((2-methoxy-4-(4-methylpiperazin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)methyl)phenyl)acrylamide
分子名称: N-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide, Tyrosine-protein kinase JAK3
著者McNally, R, Tan, L, Gray, N.S, Eck, M.J.
登録日2015-03-26
公開日2016-02-10
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Development of Selective Covalent Janus Kinase 3 Inhibitors.
J.Med.Chem., 58, 2015

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件を2024-06-12に公開中

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