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PDB: 1 件

8CJ7
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HDAC6 selective degraded (difluoromethyl)-1,3,4-oxadiazole substrate inhibitor
分子名称: 6-[(5-pyridin-2-yl-1,2$l^{4},3,4-tetrazacyclopenta-1,3-dien-2-yl)methyl]pyridine-3-carbohydrazide, Histone deacetylase 6, IODIDE ION, ...
著者Sandmark, J, Ek, M, Ripa, L.
登録日2023-02-12
公開日2023-10-18
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献Selective and Bioavailable HDAC6 2-(Difluoromethyl)-1,3,4-oxadiazole Substrate Inhibitors and Modeling of Their Bioactivation Mechanism.
J.Med.Chem., 66, 2023

221051

件を2024-06-12に公開中

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