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PDB: 2 件

8P05
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BU of 8p05 by Molmil
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with Leucettinib-92
分子名称: (4~{Z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{H}-imidazol-5-one, Casein kinase II subunit alpha, SULFATE ION
著者Kraemer, A, Meijer, L, Knapp, S, Structural Genomics Consortium (SGC)
登録日2023-05-09
公開日2023-05-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Leucettinibs, a Class of DYRK/CLK Kinase Inhibitors Inspired by the Marine Sponge Natural Product Leucettamine B.
J.Med.Chem., 66, 2023
8P04
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BU of 8p04 by Molmil
Crystal structure of human CLK1 in complex with Leucettinib-92
分子名称: (4~{Z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{H}-imidazol-5-one, Dual specificity protein kinase CLK1
著者Kraemer, A, Schroeder, M, Meijer, L, Knapp, S, Structural Genomics Consortium (SGC)
登録日2023-05-09
公開日2023-05-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Leucettinibs, a Class of DYRK/CLK Kinase Inhibitors Inspired by the Marine Sponge Natural Product Leucettamine B.
J.Med.Chem., 66, 2023

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件を2024-10-16に公開中

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