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PDB: 1 件

8BPY
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X-RAY STRUCTURE OF PDE9A IN COMPLEX WITH Inhibitor 13A
分子名称: (8~{S})-6-[2-(2,3-dihydroindol-1-yl)-2-oxidanylidene-ethyl]-4-(4-methylphenyl)-2-oxidanylidene-8-propyl-1,5,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile, High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A, MAGNESIUM ION, ...
著者Steuber, H.
登録日2022-11-18
公開日2022-12-28
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献BAY-7081: A Potent, Selective, and Orally Bioavailable Cyanopyridone-Based PDE9A Inhibitor.
J.Med.Chem., 65, 2022

222415

件を2024-07-10に公開中

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