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PDB: 2 件

7Q3F
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BU of 7q3f by Molmil
Bromodomain-containing 4 BD1 in complex with the inhibitor CRCM5484
分子名称: 2-[[11-ethanoyl-4-(furan-2-ylmethyl)-3-oxidanylidene-8-thia-4,6,11-triazatricyclo[7.4.0.0^{2,7}]trideca-1(9),2(7),5-trien-5-yl]sulfanyl]-~{N}-(2-methylpyridin-3-yl)ethanamide, Bromodomain-containing protein 4
著者Carrasco, K, Betzi, S, Morelli, X.
登録日2021-10-27
公開日2022-04-20
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.21 Å)
主引用文献CRCM5484: A BET-BDII Selective Compound with Differential Anti-leukemic Drug Modulation
J.Med.Chem., 65, 2022
7Q5O
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BU of 7q5o by Molmil
Bromodomain-containing 2 BD2 in complex with the inhibitor CRCM5484
分子名称: 1,2-ETHANEDIOL, 2-[[11-ethanoyl-4-(furan-2-ylmethyl)-3-oxidanylidene-8-thia-4,6,11-triazatricyclo[7.4.0.0^{2,7}]trideca-1(9),2(7),5-trien-5-yl]sulfanyl]-~{N}-(2-methylpyridin-3-yl)ethanamide, Bromodomain-containing protein 2
著者Carrasco, K, Betzi, S, Morelli, X.
登録日2021-11-04
公開日2022-04-20
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.519 Å)
主引用文献CRCM5484: A BET-BDII Selective Compound with Differential Anti-leukemic Drug Modulation
J.Med.Chem., 65, 2022

238582

件を2025-07-09に公開中

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