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PDB: 1 件

5V71
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KRAS G12C in bound to quinazoline based switch II pocket (SWIIP) binder
分子名称: 1-{4-[6-chloro-7-(2-fluorophenyl)quinazolin-4-yl]piperazin-1-yl}propan-1-one, GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, ...
著者Westover, K, Lu, J.
登録日2017-03-17
公開日2017-08-23
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.228 Å)
主引用文献KRAS G12C Drug Development: Discrimination between Switch II Pocket Configurations Using Hydrogen/Deuterium-Exchange Mass Spectrometry.
Structure, 25, 2017

222624

件を2024-07-17に公開中

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