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PDB: 4 件

8EGD
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BU of 8egd by Molmil
Branched chain ketoacid dehydrogenase kinase in complex with inhibitor
分子名称: 5-(4-methoxyphenyl)-1H-tetrazole, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Liu, S.
登録日2022-09-12
公開日2023-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.047 Å)
主引用文献Structural studies identify angiotensin II receptor blocker-like compounds as branched-chain ketoacid dehydrogenase kinase inhibitors.
J.Biol.Chem., 299, 2023
8EGQ
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BU of 8egq by Molmil
Branched chain ketoacid dehydrogenase kinase complexes
分子名称: (2S)-2-ethyl-4-{[(2'M)-2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4-yl]methyl}-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazine, ADENOSINE-5'-DIPHOSPHATE, SULFATE ION, ...
著者Liu, S.
登録日2022-09-13
公開日2023-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.955 Å)
主引用文献Structural studies identify angiotensin II receptor blocker-like compounds as branched-chain ketoacid dehydrogenase kinase inhibitors.
J.Biol.Chem., 299, 2023
8EGF
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BU of 8egf by Molmil
Branched chain ketoacid dehydrogenase kinase in complex with inhibitor
分子名称: (5P)-5-(4'-methyl[1,1'-biphenyl]-2-yl)-1H-tetrazole, ADENOSINE-5'-DIPHOSPHATE, POTASSIUM ION, ...
著者Liu, S.
登録日2022-09-12
公開日2023-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structural studies identify angiotensin II receptor blocker-like compounds as branched-chain ketoacid dehydrogenase kinase inhibitors.
J.Biol.Chem., 299, 2023
8EGU
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BU of 8egu by Molmil
Branched chain ketoacid dehydrogenase kinase complexes
分子名称: (2~{S})-3-methyl-2-[pentanoyl-[[4-[2-(2~{H}-1,2,3,4-tetrazol-5-yl)phenyl]phenyl]methyl]amino]butanoic acid, ADENOSINE-5'-DIPHOSPHATE, SULFATE ION, ...
著者Liu, S.
登録日2022-09-13
公開日2023-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.923 Å)
主引用文献Structural studies identify angiotensin II receptor blocker-like compounds as branched-chain ketoacid dehydrogenase kinase inhibitors.
J.Biol.Chem., 299, 2023

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件を2024-07-17に公開中

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