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PDB: 1 件

8W2L
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TRPM7 structure in complex with anticancer agent CCT128930 in closed state
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-[2-[(1~{S},2~{S},4~{S},5'~{R},6~{R},7~{S},8~{R},9~{S},12~{S},13~{R},16~{S})-5',7,9,13-tetramethylspiro[5-oxapentacyclo[10.8.0.0^{2,9}.0^{4,8}.0^{13,18}]icos-18-ene-6,2'-oxane]-16-yl]oxyethyl]propane-1,3-diol, 4-(4-chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-aminium, ...
著者Nadezhdin, K.D, Sobolevsky, A.I.
登録日2024-02-20
公開日2024-04-17
最終更新日2024-04-24
実験手法ELECTRON MICROSCOPY (2.45 Å)
主引用文献Structural basis of selective TRPM7 inhibition by the anticancer agent CCT128930.
Cell Rep, 43, 2024

221051

件を2024-06-12に公開中

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