7P2L
| thermostabilised 7TM domain of human mGlu5 receptor bound to photoswitchable ligand alloswitch-1 | 分子名称: | 2-chloranyl-~{N}-[2-methoxy-4-[(~{E})-pyridin-2-yldiazenyl]phenyl]benzamide, Metabotropic glutamate receptor 5,Endolysin,Metabotropic glutamate receptor 5 | 著者 | Huang, C.Y, Vinothkumar, K.R, Lebon, G. | 登録日 | 2021-07-06 | 公開日 | 2021-09-08 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.54 Å) | 主引用文献 | Agonists and allosteric modulators promote signaling from different metabotropic glutamate receptor 5 conformations. Cell Rep, 36, 2021
|
|
7FD9
| Thermostabilised full length human mGluR5-5M with orthosteric antagonist, LY341495 | 分子名称: | 2-[(1S,2S)-2-carboxycyclopropyl]-3-(9H-xanthen-9-yl)-D-alanine, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 5 | 著者 | Vinothkumar, K.R, Cannone, G, Lebon, G. | 登録日 | 2021-07-16 | 公開日 | 2021-09-08 | 最終更新日 | 2021-10-13 | 実験手法 | ELECTRON MICROSCOPY (4 Å) | 主引用文献 | Agonists and allosteric modulators promote signaling from different metabotropic glutamate receptor 5 conformations. Cell Rep, 36, 2021
|
|
7FD8
| Thermostabilised full length human mGluR5-5M bound with L-quisqualic acid | 分子名称: | (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL HEMISUCCINATE, ... | 著者 | Vinothkumar, K.R, Cannone, G, Lebon, G. | 登録日 | 2021-07-16 | 公開日 | 2021-09-08 | 最終更新日 | 2021-10-13 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Agonists and allosteric modulators promote signaling from different metabotropic glutamate receptor 5 conformations. Cell Rep, 36, 2021
|
|