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PDB: 1 件

6E4A
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BU of 6e4a by Molmil
Crystal structure of human BRD4(1) in complex with CN750
分子名称: 5-(4-{[(3-chlorophenyl)methyl]amino}-2-{4-[2-(dimethylamino)ethyl]piperazin-1-yl}quinazolin-6-yl)-1-methylpyridin-2(1H)-one, Bromodomain-containing protein 4, GLYCEROL
著者Fontano, E, White, A, Lakshminarasimhan, D, Suto, R.K.
登録日2018-07-17
公開日2018-09-12
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.26 Å)
主引用文献Discovery and lead identification of quinazoline-based BRD4 inhibitors.
Bioorg. Med. Chem. Lett., 28, 2018

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件を2024-07-24に公開中

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