PDB クエリの検索結果 - 日本蛋白質構造データバンク

PDB: 2 件

Crystal Structure of BRD4 with QC4956
分子名称:	4-[5-(ethylsulfonyl)-2-methoxyphenyl]-2-methyl-6-(1-methyl-1H-pyrazol-4-yl)isoquinolin-1(2H)-one, Bromodomain-containing protein 4
著者	Hosfield, D.J.
登録日	2018-02-28
公開日	2018-05-02
最終更新日	2023-10-04
実験手法	X-RAY DIFFRACTION (1.72 Å)
主引用文献	Design, synthesis and biological evaluation of novel 4-phenylisoquinolinone BET bromodomain inhibitors. Bioorg. Med. Chem. Lett., 28, 2018

Crystal Structure of BRD4 with QC4956
分子名称:	Bromodomain-containing protein 4, N-{3-[2-methyl-6-(1-methyl-1H-pyrazol-4-yl)-1-oxo-1,2-dihydroisoquinolin-4-yl]phenyl}methanesulfonamide
著者	Hosfield, D.J.
登録日	2018-02-28
公開日	2018-05-02
最終更新日	2023-10-04
実験手法	X-RAY DIFFRACTION (1.62 Å)
主引用文献	Design, synthesis and biological evaluation of novel 4-phenylisoquinolinone BET bromodomain inhibitors. Bioorg. Med. Chem. Lett., 28, 2018