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PDB: 1 件

4WLB
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BU of 4wlb by Molmil
Crystal structure of RORc in complex with a partial inverse agonist compound
分子名称: L(+)-TARTARIC ACID, N-(4-fluorobenzyl)-N-(2-methylpropyl)-6-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyridine-3-sulfonamide, Nuclear receptor ROR-gamma, ...
著者Boenig, G, Hymowitz, S.G, Kiefer, J.R.
登録日2014-10-07
公開日2014-11-12
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.702 Å)
主引用文献A reversed sulfonamide series of selective RORc inverse agonists.
Bioorg.Med.Chem.Lett., 24, 2014

224201

件を2024-08-28に公開中

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