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PDB: 1 件

3MJW
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PI3 Kinase gamma with a benzofuranone inhibitor
分子名称: (2Z)-4,6-dihydroxy-2-[(8-methoxy-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)methylidene]-1-benzofuran-3(2H)-one, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
著者Bard, J, Svenson, K.
登録日2010-04-13
公開日2010-06-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.87 Å)
主引用文献5-Ureidobenzofuranone indoles as potent and efficacious inhibitors of PI3 kinase-alpha and mTOR for the treatment of breast cancer.
Bioorg.Med.Chem.Lett., 20, 2010

221051

件を2024-06-12に公開中

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