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PDB: 2 件

5V7T
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BU of 5v7t by Molmil
crystal structure of PARP14 bound to N-{4-[4-(diphenylmethoxy)piperidin-1-yl]butyl}[1,2,4]triazolo[4,3-b]pyridazin-6-amine inhibitor
分子名称: N-{4-[4-(diphenylmethoxy)piperidin-1-yl]butyl}[1,2,4]triazolo[4,3-b]pyridazin-6-amine, Poly [ADP-ribose] polymerase 14
著者saikatendu, k.s, Hirozane, M.
登録日2017-03-20
公開日2017-05-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Identification of PARP14 inhibitors using novel methods for detecting auto-ribosylation.
Biochem. Biophys. Res. Commun., 486, 2017
5V7W
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BU of 5v7w by Molmil
Crystal structure of human PARP14 bound to 2-{[(1-methylpiperidin-4-yl)methyl]amino}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one inhibitor
分子名称: 2-{[(1-methylpiperidin-4-yl)methyl]amino}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one, Poly [ADP-ribose] polymerase 14
著者saikatendu, k.s, Hirozane, M.
登録日2017-03-20
公開日2017-05-10
最終更新日2018-11-14
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Identification of PARP14 inhibitors using novel methods for detecting auto-ribosylation.
Biochem. Biophys. Res. Commun., 486, 2017

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件を2024-07-10に公開中

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