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PDB: 4 件

6QUU
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BU of 6quu by Molmil
Crystal Structure of KRAS-G12D in complex with GMP-PCP
分子名称: GTPase KRas, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER
著者Fischer, G, Kessler, D, Muellauer, B, Wolkerstorfer, B.
登録日2019-02-28
公開日2019-07-31
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.477 Å)
主引用文献KRAS Binders Hidden in Nature.
Chemistry, 25, 2019
6QUV
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BU of 6quv by Molmil
Crystal Structure of KRAS-G12D in complex with GMP-PCP and compound 15R
分子名称: (6~{a}~{R},11~{b}~{S})-6~{a}-(1,4-dimethylpiperidin-4-yl)-7,11~{b}-dihydro-6~{H}-indolo[2,3-c]isoquinolin-5-one, GTPase KRas, MAGNESIUM ION, ...
著者Fischer, G, Kessler, D, Muellauer, B, Wolkerstorfer, B.
登録日2019-02-28
公開日2019-07-31
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.475 Å)
主引用文献KRAS Binders Hidden in Nature.
Chemistry, 25, 2019
6QUX
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BU of 6qux by Molmil
Crystal Structure of KRAS-G12D in Complex with Natural Product-Like Compound 15
分子名称: (6~{a}~{R},11~{b}~{S})-6~{a}-(1,4-dimethylpiperidin-4-yl)-7,11~{b}-dihydro-6~{H}-indolo[2,3-c]isoquinolin-5-one, 1,2-ETHANEDIOL, GTPase KRas, ...
著者Fischer, G, Kessler, D, Muellauer, B, Wolkerstorfer, B.
登録日2019-02-28
公開日2019-07-31
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.62 Å)
主引用文献KRAS Binders Hidden in Nature.
Chemistry, 25, 2019
6QUW
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BU of 6quw by Molmil
Crystal Structure of KRAS-G12D in Complex with Natural Product-Like Compound 9b
分子名称: (3~{a}~{R},8~{b}~{S})-2,2,3~{a},8~{b}-tetramethyl-3,4-dihydro-1~{H}-pyrrolo[2,3-b]indole, GTPase KRas, MAGNESIUM ION, ...
著者Fischer, G, Kessler, D, Muellauer, B, Wolkerstorfer, B.
登録日2019-02-28
公開日2019-07-31
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.242 Å)
主引用文献KRAS Binders Hidden in Nature.
Chemistry, 25, 2019

221051

件を2024-06-12に公開中

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