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PDB: 4 件

4MNV
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BU of 4mnv by Molmil
Crystal structure of bicyclic peptide UK729 bound as an acyl-enzyme intermediate to urokinase-type plasminogen activator (uPA)
分子名称: 1,3,5-tris(bromomethyl)benzene, ACETATE ION, GLYCEROL, ...
著者Chen, S, Pojer, F, Heinis, C.
登録日2013-09-11
公開日2014-02-05
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Peptide ligands stabilized by small molecules.
Angew.Chem.Int.Ed.Engl., 53, 2014
4MNX
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BU of 4mnx by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK811
分子名称: 1,1',1''-(1,3,5-triazinane-1,3,5-triyl)tripropan-1-one, GLYCEROL, SULFATE ION, ...
著者Chen, S, Pojer, F, Heinis, C.
登録日2013-09-11
公開日2014-02-05
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Peptide ligands stabilized by small molecules.
Angew.Chem.Int.Ed.Engl., 53, 2014
4MNY
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BU of 4mny by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK903
分子名称: ACETATE ION, GLYCEROL, N,N',N''-benzene-1,3,5-triyltris(2-bromoacetamide), ...
著者Chen, S, Pojer, F, Heinis, C.
登録日2013-09-11
公開日2014-02-05
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Peptide ligands stabilized by small molecules.
Angew.Chem.Int.Ed.Engl., 53, 2014
4MNW
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BU of 4mnw by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK749
分子名称: 1,3,5-tris(bromomethyl)benzene, ACETATE ION, GLYCEROL, ...
著者Chen, S, Pojer, F, Heinis, C.
登録日2013-09-11
公開日2014-02-05
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Peptide ligands stabilized by small molecules.
Angew.Chem.Int.Ed.Engl., 53, 2014

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件を2024-07-24に公開中

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