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8FPZ
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BU of 8fpz by Molmil
LBD conformation 3 (LBDconf3) of GluA2 flip Q isoform of AMPA receptor in complex with gain-of-function TARP gamma-2, with 500mM NaCl, 330uM CTZ, and 100mM glutamate (Open-Na610)
Descriptor: CYCLOTHIAZIDE, GLUTAMIC ACID, Glutamate receptor 2
Authors:Nakagawa, T.
Deposit date:2023-01-05
Release date:2024-03-06
Last modified:2024-05-01
Method:ELECTRON MICROSCOPY (3.01 Å)
Cite:The open gate of the AMPA receptor forms a Ca 2+ binding site critical in regulating ion transport.
Nat.Struct.Mol.Biol., 31, 2024
8FQA
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BU of 8fqa by Molmil
LBD conformation 2 (LBDconf2) of GluA2 flip Q isoform of AMPA receptor in complex with gain-of-function TARP gamma2, with 140mM NMDG, 330uM CTZ, and 100mM L-glutamate (Open-Na110)
Descriptor: CYCLOTHIAZIDE, GLUTAMIC ACID, Glutamate receptor 2
Authors:Nakagawa, T.
Deposit date:2023-01-05
Release date:2024-03-06
Last modified:2024-05-01
Method:ELECTRON MICROSCOPY (3.35 Å)
Cite:The open gate of the AMPA receptor forms a Ca 2+ binding site critical in regulating ion transport.
Nat.Struct.Mol.Biol., 31, 2024
8GPR
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BU of 8gpr by Molmil
GluK1-1a receptor captured in the desensitized state
Descriptor: Glutamate receptor
Authors:Dhingra, S, Kumar, J.
Deposit date:2022-08-26
Release date:2023-08-30
Last modified:2024-03-13
Method:ELECTRON MICROSCOPY (8.2 Å)
Cite:Functional Implications of the Exon 9 Splice Insert in GluK1 Kainate Receptors
Elife, 2023
8GC2
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BU of 8gc2 by Molmil
Domoate-bound GluK2 kainate receptor in partially-open conformation 1
Descriptor: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Bogdanovic, N, Tajima, N.
Deposit date:2023-03-01
Release date:2024-03-13
Method:ELECTRON MICROSCOPY (4.1 Å)
Cite:Structural basis for kainate receptor activation by a partial agonist
To Be Published
8GC4
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BU of 8gc4 by Molmil
Domoate-bound GluK2 kainate receptor in partially-open conformation 3
Descriptor: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Bogdanovic, N, Tajima, N.
Deposit date:2023-03-01
Release date:2024-03-13
Method:ELECTRON MICROSCOPY (3.93 Å)
Cite:Structural basis for kainate receptor activation by a partial agonist
To Be Published
8GC3
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BU of 8gc3 by Molmil
Domote-bound GluK2 kainate receptors in partially-open conformation 2
Descriptor: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Bogdanovic, N, Tajima, N.
Deposit date:2023-03-01
Release date:2024-03-13
Method:ELECTRON MICROSCOPY (3.8 Å)
Cite:Structural basis for kainate receptor activation by a partial agonist
To Be Published
8GC5
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BU of 8gc5 by Molmil
Domoate-bound GluK2 kainate receptors in non-active conformation
Descriptor: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Bogdanovic, N, Tajima, N.
Deposit date:2023-03-01
Release date:2024-03-13
Method:ELECTRON MICROSCOPY (3.93 Å)
Cite:Structural basis for kainate receptor activation by a partial agonist
To Be Published
8HDK
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BU of 8hdk by Molmil
Structure of the Rat GluN1-GluN2C NMDA receptor in complex with glycine and glutamate (minor class in symmetry)
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, ...
Authors:Zhang, M, Zhang, J, Guo, F, Li, Y, Zhu, S.
Deposit date:2022-11-04
Release date:2023-03-29
Last modified:2023-05-31
Method:ELECTRON MICROSCOPY (4.3 Å)
Cite:Distinct structure and gating mechanism in diverse NMDA receptors with GluN2C and GluN2D subunits.
Nat.Struct.Mol.Biol., 30, 2023
7F57
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BU of 7f57 by Molmil
Kainate-bound GluK2-1xNeto2 complex, at the desensitized state
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (3.8 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F56
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BU of 7f56 by Molmil
DNQX-bound GluK2-1xNeto2 complex, with asymmetric LBD
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (4.1 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F5A
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BU of 7f5a by Molmil
DNQX-bound GluK2-2xNeto2 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (6.4 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F59
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BU of 7f59 by Molmil
DNQX-bound GluK2-1xNeto2 complex
Descriptor: (1S)-2-{[{[(2R)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (4.2 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F5B
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BU of 7f5b by Molmil
LBD-TMD focused reconstruction of DNQX-bound GluK2-1xNeto2 complex
Descriptor: (1S)-2-{[{[(2R)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:He, L.L, Gao, Y.W, Li, B, Zhao, Y.
Deposit date:2021-06-21
Release date:2021-09-29
Last modified:2021-12-01
Method:ELECTRON MICROSCOPY (3.9 Å)
Cite:Kainate receptor modulation by NETO2.
Nature, 599, 2021

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PDB entries from 2024-06-12

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