5SQY
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![BU of 5sqy by Molmil](/molmil-images/mine/5sqy) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5211314110 - (S,S) isomer | Descriptor: | (1S,2S)-1-{[4-(cyclopropylcarbamamido)-1,3-benzothiazole-7-carbonyl]amino}-4-hydroxy-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.05 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SR4
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![BU of 5sr4 by Molmil](/molmil-images/mine/5sr4) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z2479779298 - (R,S) and (S,R) isomers | Descriptor: | (1R,3S)-3-[(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)amino]cyclopentan-1-ol, (1S,3R)-3-[(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)amino]cyclopentan-1-ol, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.05 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRB
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![BU of 5srb by Molmil](/molmil-images/mine/5srb) | |
5SQS
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![BU of 5sqs by Molmil](/molmil-images/mine/5sqs) | |
5SR3
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![BU of 5sr3 by Molmil](/molmil-images/mine/5sr3) | |
5SPX
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![BU of 5spx by Molmil](/molmil-images/mine/5spx) | |
5SQ3
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![BU of 5sq3 by Molmil](/molmil-images/mine/5sq3) | |
5SQF
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![BU of 5sqf by Molmil](/molmil-images/mine/5sqf) | |
5SQV
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![BU of 5sqv by Molmil](/molmil-images/mine/5sqv) | |
5SRA
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![BU of 5sra by Molmil](/molmil-images/mine/5sra) | |
5SRE
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![BU of 5sre by Molmil](/molmil-images/mine/5sre) | |
5SRL
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![BU of 5srl by Molmil](/molmil-images/mine/5srl) | |
5SRY
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![BU of 5sry by Molmil](/molmil-images/mine/5sry) | |
5SS7
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![BU of 5ss7 by Molmil](/molmil-images/mine/5ss7) | |
5SSF
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![BU of 5ssf by Molmil](/molmil-images/mine/5ssf) | |
5SQJ
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![BU of 5sqj by Molmil](/molmil-images/mine/5sqj) | |
5SSP
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![BU of 5ssp by Molmil](/molmil-images/mine/5ssp) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5459166285 - (R,R) and (S,S) isomers | Descriptor: | (1R,2R)-4-hydroxy-1-[(1H-indole-5-carbonyl)amino]-2,3-dihydro-1H-indene-2-carboxylic acid, (1S,2S)-4-hydroxy-1-[(1H-indole-5-carbonyl)amino]-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.15 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRG
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![BU of 5srg by Molmil](/molmil-images/mine/5srg) | |
5SPY
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![BU of 5spy by Molmil](/molmil-images/mine/5spy) | |
5SRJ
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![BU of 5srj by Molmil](/molmil-images/mine/5srj) | |
5SQ8
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![BU of 5sq8 by Molmil](/molmil-images/mine/5sq8) | |
5SS4
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![BU of 5ss4 by Molmil](/molmil-images/mine/5ss4) | |
5SQD
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![BU of 5sqd by Molmil](/molmil-images/mine/5sqd) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5010894382 - (R,R) and (S,S) isomers | Descriptor: | (1R,2R)-4-hydroxy-1-{[2-(hydroxymethyl)-1H-benzimidazole-5-carbonyl]amino}-2,3-dihydro-1H-indene-2-carboxylic acid, (1S,2S)-4-hydroxy-1-{[2-(hydroxymethyl)-1H-benzimidazole-5-carbonyl]amino}-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.05 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRO
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![BU of 5sro by Molmil](/molmil-images/mine/5sro) | |
5SQP
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![BU of 5sqp by Molmil](/molmil-images/mine/5sqp) | |