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8QYU
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BU of 8qyu by Molmil
Beta-cardiac myosin S1 fragment in the pre-powerstroke state complexed to Omecamtiv mecarbil
Descriptor: ADENOSINE-5'-DIPHOSPHATE, DIMETHYL SULFOXIDE, FORMIC ACID, ...
Authors:Robert-Paganin, J, Kikuti, C, Auguin, D, Rety, S, David, A, Houdusse, A.
Deposit date:2023-10-26
Release date:2023-12-13
Method:X-RAY DIFFRACTION (1.96 Å)
Cite:Omecamtiv mecarbil and Mavacamten target the same myosin pocket despite antagonistic effects in heart contraction.
Biorxiv, 2023

221051

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