5P1G
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5OZ4
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3PBZ
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![BU of 3pbz by Molmil](/molmil-images/mine/3pbz) | Endothiapepsin in complex with a fragment | Descriptor: | 4-(diethylamino)benzohydrazide, DIMETHYL SULFOXIDE, Endothiapepsin, ... | Authors: | Koester, H, Heine, A, Klebe, G. | Deposit date: | 2010-10-21 | Release date: | 2011-10-19 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.48 Å) | Cite: | A small nonrule of 3 compatible fragment library provides high hit rate of endothiapepsin crystal structures with various fragment chemotypes. J.Med.Chem., 54, 2011
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4Y4Z
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![BU of 4y4z by Molmil](/molmil-images/mine/4y4z) | Endothiapepsin in complex with fragment 73 | Descriptor: | (1Z)-N,N-diethylethanimidamide, 1,2-ETHANEDIOL, ACETATE ION, ... | Authors: | Schiebel, J, Heine, A, Klebe, G. | Deposit date: | 2015-02-11 | Release date: | 2016-03-02 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (1.48 Å) | Cite: | Crystallographic Fragment Screening of an Entire Library To Be Published
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5P0Q
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4Y43
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![BU of 4y43 by Molmil](/molmil-images/mine/4y43) | Endothiapepsin in complex with fragment 42 | Descriptor: | (1E,2E)-N,N'-di(propan-2-yl)cyclohepta-3,5-diene-1,2-diimine, 1,2-ETHANEDIOL, Endothiapepsin, ... | Authors: | Radeva, N, Uehlein, M, Weiss, M.S, Heine, A, Klebe, G. | Deposit date: | 2015-02-10 | Release date: | 2016-02-17 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (1.48 Å) | Cite: | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y3D
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5P7O
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5OYW
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![BU of 5oyw by Molmil](/molmil-images/mine/5oyw) | |
5OZX
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![BU of 5ozx by Molmil](/molmil-images/mine/5ozx) | |
5OZ5
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![BU of 5oz5 by Molmil](/molmil-images/mine/5oz5) | |
5P02
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5OYZ
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![BU of 5oyz by Molmil](/molmil-images/mine/5oyz) | |
5OZM
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![BU of 5ozm by Molmil](/molmil-images/mine/5ozm) | |
5OZH
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![BU of 5ozh by Molmil](/molmil-images/mine/5ozh) | |
5OZB
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![BU of 5ozb by Molmil](/molmil-images/mine/5ozb) | |
5P10
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![BU of 5p10 by Molmil](/molmil-images/mine/5p10) | |
5OYR
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![BU of 5oyr by Molmil](/molmil-images/mine/5oyr) | |
5P8N
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5DQ1
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![BU of 5dq1 by Molmil](/molmil-images/mine/5dq1) | Endothiapepsin in complex with fragment 34 | Descriptor: | 1,2-ETHANEDIOL, 3-[(cyclopropylamino)methyl]-8-ethylquinolin-2(1H)-one, Endothiapepsin, ... | Authors: | Radeva, N, Uehlein, M, Weiss, M, Heine, A, Klebe, G. | Deposit date: | 2015-09-14 | Release date: | 2016-09-28 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (1.489 Å) | Cite: | Crystallographic Fragment Screening of an Entire Library To Be Published
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5OZJ
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5OZN
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![BU of 5ozn by Molmil](/molmil-images/mine/5ozn) | |
5OZY
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![BU of 5ozy by Molmil](/molmil-images/mine/5ozy) | |
5P2G
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![BU of 5p2g by Molmil](/molmil-images/mine/5p2g) | |
5OZP
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![BU of 5ozp by Molmil](/molmil-images/mine/5ozp) | |