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PDB: 206 results

2JUV
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BU of 2juv by Molmil
AbaA3-DKP-insulin
Descriptor: Insulin A chain, Insulin B chain
Authors:Huang, K, Chan, S, Hua, Q, Chu, Y, Wang, R, Klaproth, B, Jia, W, Whittaker, J, De Meyts, P, Nakagawa, S.H, Steiner, D.F, Katsoyannis, P.G, Weiss, M.A.
Deposit date:2007-09-05
Release date:2007-10-16
Last modified:2021-10-20
Method:SOLUTION NMR
Cite:The A-chain of Insulin Contacts the Insert Domain of the Insulin Receptor: PHOTO-CROSS-LINKING AND MUTAGENESIS OF A DIABETES-RELATED CREVICE.
J.Biol.Chem., 282, 2007
5GSK
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BU of 5gsk by Molmil
Crystal structure of duplex DNA3 in complex with Hg(II) and Sr(II)
Descriptor: DNA (5'-D(*GP*GP*TP*CP*GP*TP*CP*C)-3'), MERCURY (II) ION, STRONTIUM ION
Authors:Liu, H.H, Wang, R, Yao, Q.Q, Cheng, Y.Q, Yang, C, Luo, Q, Wu, B.X, Li, J.X, Ma, J.B, Sheng, J, Gan, J.H.
Deposit date:2016-08-16
Release date:2017-02-08
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (1.05 Å)
Cite:Flexibility and stabilization of HgII-mediated C:T and T:T base pairs in DNA duplex
Nucleic Acids Res., 45, 2017
5TOE
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BU of 5toe by Molmil
Pim-1 kinase in complex with a 7-azaindole
Descriptor: 2-[4-(piperazin-1-yl)phenyl]-1H-pyrrolo[2,3-b]pyridine-4-carbonitrile, Serine/threonine-protein kinase pim-1
Authors:Mclean, L, Mechin, I, Zhang, Y, Wang, R, Batchelor, J.D.
Deposit date:2016-10-17
Release date:2017-10-11
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.301 Å)
Cite:Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors - Part I.
Bioorg. Med. Chem. Lett., 27, 2017
5TEX
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BU of 5tex by Molmil
Pim-1 kinase in complex with a 7-azaindole
Descriptor: (4-{4-chloro-1-methyl-2-[4-(piperazin-1-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl}phenyl)methanol, IMIDAZOLE, Serine/threonine-protein kinase pim-1
Authors:Mechin, I, Wang, R, Batchelor, J.D, McLean, L.
Deposit date:2016-09-23
Release date:2017-10-11
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.149 Å)
Cite:Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors - Part I.
Bioorg. Med. Chem. Lett., 27, 2017
5TUR
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BU of 5tur by Molmil
Pim-1 kinase in complex with a 7-azaindole
Descriptor: 1-methyl-2-[4-(piperazin-1-yl)phenyl]-1H-pyrrolo[2,3-b]pyridine-4-carbonitrile, Serine/threonine-protein kinase pim-1
Authors:Mechin, I, Zhang, Y, Wang, R, Batchelor, J.D, Mclean, L.
Deposit date:2016-11-07
Release date:2017-10-11
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.948 Å)
Cite:Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors - Part I.
Bioorg. Med. Chem. Lett., 27, 2017
5TEL
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BU of 5tel by Molmil
Pim-1 kinase in complex with a 7-azaindole
Descriptor: 4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1H-indol-3-yl}-1H-pyrrolo[2,3-b]pyridine, IMIDAZOLE, Serine/threonine-protein kinase pim-1
Authors:Mechin, I, Wang, R, Batchelor, J.D.
Deposit date:2016-09-22
Release date:2017-10-11
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.214 Å)
Cite:Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors - Part I.
Bioorg. Med. Chem. Lett., 27, 2017

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