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PDB: 29 件

4YUS
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BU of 4yus by Molmil
Crystal structure of photoactivated adenylyl cyclase of a cyanobacteriaOscillatoria acuminata in hexagonal form
分子名称: FLAVIN MONONUCLEOTIDE, Family 3 adenylate cyclase
著者Park, S.-Y, Ohki, M, Sugiyama, K, Kawai, F, Iseki, M.
登録日2015-03-19
公開日2016-06-01
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural insight into photoactivation of an adenylate cyclase from a photosynthetic cyanobacterium
Proc.Natl.Acad.Sci.USA, 113, 2016
4YUT
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BU of 4yut by Molmil
Crystal structure of photoactivated adenylyl cyclase of a cyanobacteriaOscillatoria acuminata in orthorhombic form
分子名称: FLAVIN MONONUCLEOTIDE, Family 3 adenylate cyclase
著者Park, S.-Y, Ohki, M, Sugiyama, K, Kawai, F, Iseki, M.
登録日2015-03-19
公開日2016-06-01
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural insight into photoactivation of an adenylate cyclase from a photosynthetic cyanobacterium
Proc.Natl.Acad.Sci.USA, 113, 2016
3WX7
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BU of 3wx7 by Molmil
Crystal structure of COD
分子名称: ACETATE ION, CALCIUM ION, Chitin oligosaccharide deacetylase, ...
著者Park, S.-Y, Sugiyama, K, Hirano, T, Nishio, T.
登録日2014-07-18
公開日2014-12-03
最終更新日2019-04-03
実験手法X-RAY DIFFRACTION (1.349 Å)
主引用文献Structure-based analysis of domain function of chitin oligosaccharide deacetylase from Vibrio parahaemolyticus.
FEBS Lett., 589, 2015
5X02
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BU of 5x02 by Molmil
Crystal structure of the FLT3 kinase domain bound to the inhibitor FF-10101
分子名称: N-[(2S)-1-[5-[2-[(4-cyanophenyl)amino]-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxidanylidene-propan-2-yl]-4-(dimethylamino)-N-methyl-but-2-enamide, Receptor-type tyrosine-protein kinase FLT3, SULFATE ION
著者Fujikawa, N, Hirano, D, Takasaki, M, Terada, D, Hagiwara, S, Park, S.-Y, Sugiyama, K.
登録日2017-01-19
公開日2018-01-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.401 Å)
主引用文献A novel irreversible FLT3 inhibitor, FF-10101, shows excellent efficacy against AML cells withFLT3mutations.
Blood, 131, 2018
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件を2024-05-29に公開中

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