3WZU
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![BU of 3wzu by Molmil](/molmil-images/mine/3wzu) | THE STRUCTURE OF MAP2K7 IN COMPLEX WITH 5Z-7-oxozeaenol | 分子名称: | (3S,5Z,8S,9S,11E)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1H-2-benzoxacyclotetradecine-1,7(8H)-dione, Dual specificity mitogen-activated protein kinase kinase 7 | 著者 | Sogabe, Y, Hashimoto, Y, Matsumoto, T, Kinoshita, T. | 登録日 | 2014-10-07 | 公開日 | 2015-01-14 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.01 Å) | 主引用文献 | 5Z-7-Oxozeaenol covalently binds to MAP2K7 at Cys218 in an unprecedented manner. Bioorg.Med.Chem.Lett., 25, 2015
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5B2L
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![BU of 5b2l by Molmil](/molmil-images/mine/5b2l) | A crucial role of Cys218 in the stabilization of an unprecedented auto-inhibition form of MAP2K7 | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Dual specificity mitogen-activated protein kinase kinase 7, GLYCEROL | 著者 | Sogabe, Y, Hashimoto, T, Matsumoto, T, Kirii, Y, Sawa, M, Kinoshita, T. | 登録日 | 2016-01-19 | 公開日 | 2016-04-06 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | A crucial role of Cys218 in configuring an unprecedented auto-inhibition form of MAP2K7 Biochem.Biophys.Res.Commun., 473, 2016
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5B2K
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![BU of 5b2k by Molmil](/molmil-images/mine/5b2k) | A crucial role of Cys218 in the stabilization of an unprecedented auto-inhibition form of MAP2K7 | 分子名称: | Dual specificity mitogen-activated protein kinase kinase 7 | 著者 | Sogabe, Y, Hashimoto, T, Matsumoto, T, Kirii, Y, Sawa, M, Kinoshita, T. | 登録日 | 2016-01-19 | 公開日 | 2016-04-06 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | A crucial role of Cys218 in configuring an unprecedented auto-inhibition form of MAP2K7 Biochem.Biophys.Res.Commun., 473, 2016
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5B2M
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![BU of 5b2m by Molmil](/molmil-images/mine/5b2m) | A crucial role of Cys218 in the stabilization of an unprecedented auto-inhibition form of MAP2K7 | 分子名称: | Dual specificity mitogen-activated protein kinase kinase 7 | 著者 | Sogabe, Y, Hashimoto, T, Matsumoto, T, Kirii, Y, Sawa, M, Kinoshita, T. | 登録日 | 2016-01-19 | 公開日 | 2016-04-06 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.06 Å) | 主引用文献 | A crucial role of Cys218 in configuring an unprecedented auto-inhibition form of MAP2K7 Biochem.Biophys.Res.Commun., 473, 2016
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3A72
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![BU of 3a72 by Molmil](/molmil-images/mine/3a72) | |
3A71
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![BU of 3a71 by Molmil](/molmil-images/mine/3a71) | |
3WAR
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![BU of 3war by Molmil](/molmil-images/mine/3war) | Crystal structure of human CK2a | 分子名称: | 1,2-ETHANEDIOL, Casein kinase II subunit alpha, NICOTINIC ACID | 著者 | Kinoshita, T, Nakaniwa, T, Sekiguchi, Y, Sogabe, Y, Sakurai, A, Nakamura, S, Nakanishi, I. | 登録日 | 2013-05-07 | 公開日 | 2013-10-30 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.04 Å) | 主引用文献 | Crystal structure of human CK2 alpha at 1.06 angstrom resolution J.SYNCHROTRON RADIAT., 20, 2013
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3WOW
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![BU of 3wow by Molmil](/molmil-images/mine/3wow) | Crystal structure of human CK2a with AMPPNP | 分子名称: | 1,2-ETHANEDIOL, Casein kinase II subunit alpha, MAGNESIUM ION, ... | 著者 | Kinoshita, T, Nakaniwa, T, Sekiguchi, Y, Sogabe, Y, Sakurai, A, Nakamura, S, Nakanishi, I, Shimada, K, Tanaka, M. | 登録日 | 2014-01-06 | 公開日 | 2015-02-04 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | A hydrophobic residue divergence of CK2a contribute to a species-dependent variation for apigenin binding mode but not for an ATP analogue To be Published
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5Y90
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![BU of 5y90 by Molmil](/molmil-images/mine/5y90) | MAP2K7 mutant -C218S | 分子名称: | Dual specificity mitogen-activated protein kinase kinase 7, GLYCEROL | 著者 | Kinoshita, T, Hashimoto, T, Sogabe, Y, Matsumoto, T, Sawa, M, Fukada, H. | 登録日 | 2017-08-22 | 公開日 | 2017-10-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | High-resolution structure discloses the potential for allosteric regulation of mitogen-activated protein kinase kinase 7 Biochem. Biophys. Res. Commun., 493, 2017
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